Cedazuridine

Cedazuridine

SCHEMBL172256

O=C1N[C@H](O)CCN1[C@@H]1O[C@H](CO)[C@@H](O)C1(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

CDA

The experimentally established mechanism targets of Cedazuridine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CDA known ✓ P32320 11/20 1.00
PDE4D Q08499 1/20 0.43
PDE3A Q14432 1/20 0.43
SLC29A1 Q99808 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cedazuridine SCHEMBL170217 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL13828324 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL10070522 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL10069553 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL23227281 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL24807958 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL10070136 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL25286013 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL19965745 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1
Cedazuridine SCHEMBL19965746 1.00 CDA (1.00) CDAPDE4DPDE3ASLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 441 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4743074-A1 METHODS OF TREATING HEMATOLOGIC CANCER Foghorn Therapeutics Inc. (US) 2026-05-20 EP claimed
US-20260124190-A1 METHOD FOR TREATING A DISEASE OR CONDITION USING A PYRAZOLE COMPOUND OR FORMULATION THEREOF RIGEL PHARMACEUTICALS, INC. (US) 2026-05-07 US claimed
EP-4727596-A2 ANTIBODY-DRUG CONJUGATES AND LINKERS AND METHODS OF USE THEREOF Ohio State Innovation Foundation (US) 2026-04-22 EP claimed
EP-4709378-A1 COMPOUNDS FOR NOS-RELATED CANCERS AND METHODS OF USE Yissum Research Development Company of the Hebrew University of Jerusalem Ltd. (IL) 2026-03-18 EP claimed
EP-4704834-A1 RESPONSE-BASED DOSING FOR TREATING CANCER WITH A HYPOMETHYLATING AGENT AND CEDAZURIDINE Taiho Pharmaceutical Co., Ltd. (JP) 2026-03-11 EP claimed
US-12514866-B2 Method for treating cancer NATIONAL TAIWAN UNIVERSITY (TW) 2026-01-06 US claimed
US-20260000697-A1 COMBINATION FORMULATION OF CEDAZURIDINE OTSUKA PHARMA CO LTD (JP) 2026-01-01 US claimed
EP-4663205-A1 POLYMER-DRUG CONJUGATE, INTERMEDIATE THEREOF, AND USE THEREOF Shanghai Best-Link Bioscience, LLC (CN) 2025-12-17 EP claimed
US-20250288687-A1 COMBINATION OF ANTIBODY-DRUG CONJUGATES AND DNMT INHIBITORS DAIICHI SANKYO COMPANY, LIMITED (JP) 2025-09-18 US claimed
US-20250255977-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF SHANGHAI BEST-LINK BIOSCIENCE, LLC (CN) 2025-08-14 US claimed
US-11660310-B2 Low dose combination CDA substrate drug/cedazuridine with extended administration OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2023-05-30 US claimed
WO-2023078464-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF 上海弼领生物技术有限公司 2023-05-11 WO claimed
US-20230089147-A1 COMBINATION DECITABINE AND CEDAZURIDINE SOLID ORAL DOSAGE FORMS TAIHO PHARMACEUTICAL CO., LTD. (JP) 2023-03-23 US claimed
CN-115381939-A Pharmaceutical composition for treating Hodgkin lymphoma and application thereof 深圳微芯生物科技股份有限公司 2022-11-25 CN claimed
WO-2022221304-A1 CO-INHIBITION OF CD47/SIRPα BINDING AND NEDD8-ACTIVATING ENZYME E1 REGULATORY SUBUNIT FOR THE TREATMENT OF CANCER GILEAD SCIENCES, INC. (US) 2022-10-20 WO claimed
WO-2022204126-A1 TREATMENT OF RNA VIRUS INFECTION WITH A CYTIDINE DEAMINASE INHIBITOR THE CLEVELAND CLINIC FOUNDATION (US) 2022-09-29 WO claimed
US-20220288047-A1 METHOD FOR TREATING A DISEASE OR CONDITION USING A PYRAZOLE COMPOUND OR FORMULATION THEREOF RIGEL PHARMACEUTICALS, INC. (US) 2022-09-15 US claimed
WO-2022187303-A1 A METHOD FOR TREATING A DISEASE OR CONDITION USING A PYRAZOLE COMPOUND OR FORMULATION THEREOF RIGEL PHARMACEUTICALS, INC. (US) 2022-09-09 WO claimed
WO-2022093930-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME FOR TREATING CANCER OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2022-05-05 WO claimed
US-20220110958-A1 LOW DOSE COMBINATION CDA SUBSTRATE DRUG/CEDAZURIDINE WITH EXTENDED ADMINISTRATION TAIHO PHARMACEUTICAL CO., LTD. (JP) 2022-04-14 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220288047-A1 METHOD FOR TREATING A DISEASE OR CONDITION USING A PYRAZOLE COMPOUND OR FORMULATION THEREOF MCL1, IL5, MALT1 CDA 2213/4885PDE4D 3988/4885PDE3A 1818/4885
US-20260000697-A1 COMBINATION FORMULATION OF CEDAZURIDINE DCTD, EZH2, DUT CDA 4/4885PDE4D 136/4885PDE3A 228/4885
US-20220110958-A1 LOW DOSE COMBINATION CDA SUBSTRATE DRUG/CEDAZURIDINE WITH EXTENDED ADMINISTRATION CDA, DNMT1, DUT CDA 1/4885PDE4D 2182/4885PDE3A 2945/4885
US-20250255977-A1 EPSILON-POLY-L-LYSINE-BASED DRUG CONJUGATE, INTERMEDIATE THEREOF, AND APPLICATION THEREOF SLC7A1, KARS1, LNPEP CDA 1286/4885PDE4D 3249/4885PDE3A 2974/4885
US-20250288687-A1 COMBINATION OF ANTIBODY-DRUG CONJUGATES AND DNMT INHIBITORS DNMT1, DNMT3B, DNMT3A CDA 342/4885PDE4D 2399/4885PDE3A 2004/4885
US-20260124190-A1 METHOD FOR TREATING A DISEASE OR CONDITION USING A PYRAZOLE COMPOUND OR FORMULATION THEREOF IRAK2, IRAK3, IRAK1 CDA 2389/4885PDE4D 2068/4885PDE3A 2658/4885
US-20230089147-A1 COMBINATION DECITABINE AND CEDAZURIDINE SOLID ORAL DOSAGE FORMS DNMT3A, DNMT1, CDA CDA 3/4885PDE4D 464/4885PDE3A 613/4885
US-11660310-B2 Low dose combination CDA substrate drug/cedazuridine with extended administration CDA, DNMT1, DUT CDA 1/4885PDE4D 2182/4885PDE3A 2945/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.