SCHEMBL1723280

SCHEMBL1723280

Cn1cnc(S(=O)(=O)N(Cc2ccc(F)cc2)c2ccc(C(=O)O)cc2)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
POLB P06746 1/20 0.49
KCNA5 P22460 1/20 0.47
TAS2R14 Q9NYV8 5/20 0.47
PTGES O14684 5/20 0.46
ALOX5 P09917 3/20 0.46
TRPM8 Q7Z2W7 2/20 0.44
FNTA P49354 1/20 0.44
FNTB P49356 1/20 0.44
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
TP53 P04637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1722397 0.90 MEN1 (0.61) KMT2AMEN1POLBPTGESALOX5
SCHEMBL3281840 0.89 KMT2A (0.51) KMT2AMEN1TAS2R14PTGESALOX5
SCHEMBL1722971 0.83 MEN1 (0.51) KMT2AMEN1POLBTAS2R14PTGES
SCHEMBL327423 0.82 POLB (0.46) KMT2AMEN1POLBALDH1A1HPGD
SCHEMBL2212915 0.79 MEN1 (0.58) KMT2AMEN1PTGESALOX5FNTA
SCHEMBL3275416 0.78 RAB9A (0.52) KMT2AMEN1POLBFNTAFNTB
SCHEMBL1723248 0.78 MEN1 (0.55) KMT2AMEN1POLBTRPM8FNTA
SCHEMBL3279243 0.78 FNTA (0.65) KMT2AMEN1PTGESALOX5FNTA
SCHEMBL2211492 0.78 MEN1 (0.53) KMT2AMEN1POLBTAS2R14FNTA
SCHEMBL303692 0.77 LMNA (0.66) KMT2AMEN1POLBFNTAFNTB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344456-B1 NOVEL POTASSIUM CHANNEL BLOCKER JAPAN TOBACCO INC (JP) 2018-07-25 EP disclosed
US-8258138-B2 Potassium channel blockers XENTION LIMITED (GB) 2012-09-04 US disclosed
EP-2344456-A1 NOVEL POTASSIUM CHANNEL BLOCKER Xention Limited (GB) 2011-07-20 EP disclosed
US-20100087437-A1 Novel Potassium Channel Blockers XENTION LIMITED (GB) 2010-04-08 US disclosed
WO-2010023445-A1 NOVEL POTASSIUM CHANNEL BLOCKER XENTION LIMITED (GB) 2010-03-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100087437-A1 Novel Potassium Channel Blockers KCNB1, KCNJ2, KCNJ11 KMT2A 777/4885MEN1 824/4885POLB 4525/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.