SCHEMBL17243774

SCHEMBL17243774

COc1ccc(OCc2nnc([C@@H]3CCCN3C(=O)OC(C)(C)C)o2)cc1OC

nearest known ligand 0.52

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
TSHR P16473 7/20 0.49
LMNA P02545 6/20 0.49
KMT2A Q03164 4/20 0.49
MEN1 O00255 3/20 0.49
MAPT P10636 2/20 0.49
NPSR1 Q6W5P4 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
HTT P42858 1/20 0.49
GAA P10253 1/20 0.46
POLB P06746 1/20 0.46
TP53 P04637 2/20 0.45
GLA P06280 1/20 0.45
EPHA2 P29317 1/20 0.41
KDR P35968 1/20 0.41
EPHB4 P54760 1/20 0.41
FKBP1A P62942 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17243796 0.86 ALDH1A1 (0.46) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL3180503 0.83 SCD (0.43) ALDH1A1TSHRMAPTEPHA2KDR
SCHEMBL17243781 0.83 EPHA2 (0.58) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL17103763 0.81 ALDH1A1 (0.36) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL17103764 0.81 ALDH1A1 (0.36) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL15417979 0.80 FKBP1A (0.41) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL15417963 0.80 SCD (0.42) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL17243782 0.79 FKBP1A (0.41) ALDH1A1KMT2AMEN1L3MBTL1EPHA2
SCHEMBL17243786 0.79 MEN1 (0.44) ALDH1A1TSHRLMNAKMT2AMEN1
SCHEMBL17243791 0.78 MEN1 (0.42) KMT2AMEN1L3MBTL1HTTEPHA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9181229-B2 Azole derivative TAISHO PHARMACEUTICAL CO., LTD. (JP) 2015-11-10 US disclosed
US-9181229-B2 Azole derivative TAISHO PHARMACEUTICAL CO., LTD. (JP) 2015-11-10 US disclosed