SCHEMBL172440

SCHEMBL172440

Cc1ccc2nc(I)[nH]c2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.58
POLB P06746 1/20 0.58
ALDH1A1 P00352 3/20 0.56
HPGD P15428 2/20 0.56
USP2 O75604 1/20 0.56
HTT P42858 1/20 0.56
CYP1A2 P05177 1/20 0.54
PIN1 Q13526 1/20 0.54
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
GAA P10253 2/20 0.53
HSD17B10 Q99714 2/20 0.53
KDM4E B2RXH2 3/20 0.50
ADORA2A P29274 1/20 0.50
MMP2 P08253 1/20 0.49
MMP9 P14780 1/20 0.49
MMP8 P22894 1/20 0.49
MMP13 P45452 1/20 0.49
METAP2 P50579 2/20 0.49
METAP1 P53582 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22800202 0.84 KMT2A (0.44) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL29727934 0.79 ALDH1A1 (0.66) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL266609 0.79 ALDH1A1 (0.66) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL9306275 0.76 ALDH1A1 (0.61) KMT2AALDH1A1HPGDCYP1A2NPC1
SCHEMBL15947574 0.76 ALDH1A1 (0.61) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL229608 0.76 KMT2A (0.58) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL2780693 0.76 KMT2A (0.58) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL9305169 0.76 KMT2A (0.58) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL827359 0.76 KMT2A (0.58) KMT2APOLBALDH1A1HPGDUSP2
SCHEMBL2360748 0.76 PLAU (0.61) KMT2APOLBALDH1A1HPGDUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3172214-B1 2-AMINO-PYRIDO[2,3-D]PYRIMIDIN-7(8H)-ONE DERIVATIVES AS CDK INHIBITORS AND USES THEREOF SUNSHINE LAKE PHARMA CO LTD (CN) 2020-05-13 EP disclosed
WO-2014082379-A1 SPIRO RING COMPOUND AS HEPATITIS C VIRUS (HCV) INHIBITOR AND USES THEREOF FIELD OF THE INVENTION SUNSHINE LAKE PHARMA CO.,LTD. (CN) 2014-06-05 WO disclosed
WO-2013059278-A2 HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2013-04-25 WO disclosed
EP-1919891-B1 3,5-DISUBSTITUTED PYRID-2-ONES USEFUL AS INHIBITORS OF TEC FAMILY OF NON-RECEPTOR TYROSINE KINASES VERTEX PHARMA (US) 2012-03-07 EP disclosed
WO-2007062342-A1 HETEROCYCLIC CETP INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-31 WO disclosed