SCHEMBL1724657

SCHEMBL1724657

COc1cc(F)c(-c2c(C)nn(C)c2N)c(F)c1.COc1cc(F)c(C(C#N)C(C)=O)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.35
PDE10A Q9Y233 1/20 0.35
CYP1A2 P05177 2/20 0.35
GRM8 O00222 1/20 0.35
GRM7 Q14831 1/20 0.35
POLB P06746 1/20 0.34
MAPK14 Q16539 1/20 0.32
MAPT P10636 1/20 0.32
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GLA P06280 1/20 0.30
CYP2C9 P11712 1/20 0.30
HPGD P15428 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173553 0.81 PDE2A (0.47) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL158125 0.80 ALDH1A1 (0.37) ALDH1A1
SCHEMBL22609776 0.69 PTGS2 (0.40) ALDH1A1CYP2C19
SCHEMBL21342460 0.68 KMT2A (0.44) KDM4EALDH1A1HPGD
SCHEMBL671210 0.67 PTPN11 (0.37) MAPT
SCHEMBL1725188 0.66 MAPT (0.49) POLBMAPK14MAPTALDH1A1
SCHEMBL173584 0.66 PDE10A (0.47) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL17674744 0.65 MAPK14 (0.50) PDE2APDE10ACYP1A2GRM8GRM7
SCHEMBL22609734 0.64 AKR1C3 (0.36) MAPTKDM4EALDH1A1
SCHEMBL1724913 0.63 PDE2A (0.41) PDE2APDE10ACYP1A2GRM8GRM7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403834-A1 Fungicidal pyrazoles E. I. du Pont de Nemours and Company (US) 2012-01-11 EP disclosed
WO-2010101973-A1 FUNGICIDAL PYRAZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-09-10 WO disclosed