SCHEMBL172518

SCHEMBL172518

CCOc1ccn2nc(C)c(CCNC(C)=O)c2c1

nearest known ligand 0.48

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 11/20 0.48
MTNR1B P49286 9/20 0.48
ACACB O00763 3/20 0.44
NQO2 P16083 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12475741 0.66 ACACB (0.86) MTNR1AACACB
SCHEMBL126690 0.65 MTNR1A (1.00) MTNR1AMTNR1B
SCHEMBL25100769 0.65 MTNR1A (0.78) MTNR1AMTNR1BNQO2
SCHEMBL16938261 0.64 KDM4E (0.42)
SCHEMBL12001427 0.63 ACACB (0.79) MTNR1AACACB
SCHEMBL14976630 0.63 KMT2A (0.63) ACACB
SCHEMBL23099061 0.62 PRMT5 (0.45)
SCHEMBL13724706 0.62 MTNR1A (1.00) MTNR1AMTNR1B
SCHEMBL8569058 0.61 MTNR1A (0.79) MTNR1AMTNR1BNQO2
SCHEMBL255805 0.61 ACACB (1.00) ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100895-B1 TRICYCLIC COMPOUND AND MEDICAL USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2012-03-07 EP disclosed