SCHEMBL17253141

SCHEMBL17253141

FC(F)(F)Cn1ccc2cc(Br)cnc21

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 2/20 0.43
FGFR4 P22455 2/20 0.43
ENPP3 O14638 4/20 0.37
ENPP1 P22413 3/20 0.37
DGAT1 O75907 1/20 0.35
MAOB P27338 1/20 0.33
HSD17B10 Q99714 1/20 0.32
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HDAC8 Q9BY41 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857211 0.82 FGFR1 (0.43) FGFR1FGFR4ENPP3ENPP1HSD17B10
SCHEMBL22130207 0.81 DGAT1 (0.39) DGAT1
SCHEMBL17253109 0.81 DGAT1 (0.37) FGFR1FGFR4DGAT1
SCHEMBL14136876 0.78 FGFR1 (0.46) FGFR1FGFR4ENPP3ENPP1HSD17B10
SCHEMBL31126947 0.76 FGFR1 (0.44) FGFR1FGFR4ENPP3ENPP1HSD17B10
SCHEMBL23926476 0.76 ALDH1A1 (0.42) ENPP3ENPP1DGAT1MAOB
SCHEMBL15712213 0.74 FGFR1 (0.50) FGFR1FGFR4ENPP3ENPP1HDAC8
SCHEMBL7859822 0.74 HTR7 (0.42) FGFR1FGFR4ENPP3ENPP1
SCHEMBL20985874 0.73 FGFR1 (0.42) FGFR1FGFR4ENPP3ENPP1HSD17B10
SCHEMBL3560778 0.73 FGFR1 (0.42) FGFR1FGFR4ENPP3ENPP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015170775-A1 SUBSTITUTED AZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES 日産化学工業株式会社 2015-11-12 WO disclosed