SCHEMBL1725932

SCHEMBL1725932

Cc1nn(C)c(-c2ncccc2N)c1-c1ccc(F)cc1F

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
PDE10A Q9Y233 1/20 0.39
ADORA2A P29274 2/20 0.37
ADORA2B P29275 1/20 0.37
ADORA1 P30542 1/20 0.37
PDE4A P27815 1/20 0.36
GRM5 P41594 1/20 0.36
SLC34A1 Q06495 4/20 0.36
ALK Q9UM73 5/20 0.36
MAPK14 Q16539 2/20 0.36
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
NTRK2 Q16620 1/20 0.35
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1725607 0.76 MAPT (0.49) PGRNR3C2ADORA2AGRM5SLC34A1
SCHEMBL21711408 0.71 GRM5 (0.48) PGRNR3C2ADORA2AADORA2BADORA1
SCHEMBL9997510 0.70 SLC34A1 (0.42) PGRNR3C2PDE10ASLC34A1MAPK14
SCHEMBL20698315 0.69 GRM4 (0.39) SLC34A1
SCHEMBL19248544 0.69 ALDH1A1 (0.46) ADORA1MAPK14MAPK13MAPK12MAPK11
SCHEMBL30786508 0.69 PTGS2 (0.46)
SCHEMBL3488435 0.68 PGR (0.45) PGRNR3C2ADORA2AGRM5SLC34A1
SCHEMBL20697939 0.68 MAPK1 (0.41) PGRNR3C2ADORA2AADORA1SLC34A1
SCHEMBL21711491 0.67 SLC34A1 (0.47) PGRNR3C2ADORA2AADORA2BADORA1
SCHEMBL20698316 0.67 GRM4 (0.39) SLC34A1ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403834-A1 Fungicidal pyrazoles E. I. du Pont de Nemours and Company (US) 2012-01-11 EP disclosed