SCHEMBL17263229

SCHEMBL17263229

O=S(=O)(CF)N(c1ccccn1)S(=O)(=O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
HDAC1 Q13547 3/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC8 Q9BY41 1/20 0.37
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 1/20 0.34
KDM4E B2RXH2 2/20 0.33
HSD17B10 Q99714 2/20 0.33
HPGD P15428 1/20 0.33
POLQ O75417 1/20 0.33
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
MAPT P10636 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL306348 0.87 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2HDAC1HDAC6HDAC8
SCHEMBL29443546 0.87 ALDH1A1 (0.41) ALDH1A1SMN1; SMN2HDAC1HDAC6HDAC8
SCHEMBL10059165 0.76 HSP90AA1 (0.36) ALDH1A1HSD17B10TSHRKMT2ASLC6A2
SCHEMBL14307527 0.74 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2CYP2D6CYP2C19POLB
SCHEMBL15557360 0.73 ALDH1A1 (0.50) ALDH1A1SMN1; SMN2KDM4EHSD17B10LMNA
SCHEMBL11336157 0.72 POLB (0.38) ALDH1A1SMN1; SMN2HDAC1HDAC6POLB
SCHEMBL5539664 0.70 NFE2L2 (0.31)
SCHEMBL4383200 0.68 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2CYP2D6CYP2C19POLB
SCHEMBL254106 0.68 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2CYP2D6CYP2C19POLB
SCHEMBL5535038 0.68 PGK1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143018-A1 CARBOXAMIDE DERIVATIVES Novartis AG (CH) 2017-03-22 EP disclosed
WO-2015175796-A1 CARBOXAMIDE DERIVATIVES NOVARTIS AG (CH) 2015-11-19 WO disclosed