SCHEMBL1728116

SCHEMBL1728116

CC(C)(C)c1nc2c(OC(=O)NCC3CCN(CC4CCN(C(=O)c5ccc(F)cc5)CC4)CC3)cccc2[nH]1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 7/20 0.45
HTR4 Q13639 7/20 0.45
CYP3A4 P08684 1/20 0.37
GAA P10253 1/20 0.37
CYP2C9 P11712 1/20 0.37
HPGD P15428 1/20 0.37
CYP2C19 P33261 1/20 0.37
HTR2B P41595 3/20 0.37
DRD2 P14416 3/20 0.37
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
PARP1 P09874 1/20 0.37
PKM P14618 1/20 0.36
PKLR P30613 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728203 0.90 HTR3A (0.44) HTR3AHTR4PARP1
SCHEMBL1726873 0.90 HTR4 (0.48) HTR3AHTR4CYP2C9CYP2C19HTR2A
SCHEMBL828636 0.88 HTR3A (0.59) HTR3AHTR4PARP1
SCHEMBL29401326 0.88 HTR3A (0.59) HTR3AHTR4PARP1
SCHEMBL1728189 0.78 HTR4 (0.59) HTR3AHTR4HTR2AHTR2CPARP1
SCHEMBL829163 0.78 HTR4 (0.60) HTR3AHTR4PARP1
SCHEMBL29399928 0.78 HTR4 (0.60) HTR3AHTR4PARP1
SCHEMBL828465 0.76 HTR3A (0.58) HTR3AHTR4PARP1
SCHEMBL29400942 0.76 HTR3A (0.58) HTR3AHTR4PARP1
SCHEMBL829424 0.75 HTR4 (0.76) HTR3AHTR4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899324-B1 Benzimidazole-carboxamide compounds as 5-HT4 receptor agonists THERAVANCE INC (US) 2011-11-30 EP claimed