SCHEMBL1726873

SCHEMBL1726873

CC(C)(C)c1nc2c(OC(=O)NCC3CCN(CC4CCN(C(=O)c5ccccc5F)CC4)CC3)cccc2[nH]1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 10/20 0.48
HTR3A P46098 9/20 0.48
PARP1 P09874 3/20 0.40
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPK14 Q16539 1/20 0.39
PARP2 Q9UGN5 1/20 0.37
HSD11B1 P28845 1/20 0.37
AKR1C3 P42330 1/20 0.37
NPY5R Q15761 1/20 0.37
LMNA P02545 1/20 0.36
HTR7 P34969 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728116 0.90 HTR3A (0.45) HTR4HTR3APARP1HTR2AHTR2C
SCHEMBL829163 0.89 HTR4 (0.60) HTR4HTR3APARP1PARP2
SCHEMBL29399928 0.89 HTR4 (0.60) HTR4HTR3APARP1PARP2
SCHEMBL1728203 0.85 HTR3A (0.44) HTR4HTR3APARP1HSD11B1AKR1C3
SCHEMBL1728189 0.81 HTR4 (0.59) HTR4HTR3APARP1HTR2AHTR2C
SCHEMBL29401326 0.80 HTR3A (0.59) HTR4HTR3APARP1PARP2
SCHEMBL828636 0.80 HTR3A (0.59) HTR4HTR3APARP1PARP2
SCHEMBL1728218 0.79 HTR4 (0.63) HTR4HTR3APARP1CYP2C9CYP2C19
SCHEMBL829424 0.77 HTR4 (0.76) HTR4HTR3APARP1PARP2
SCHEMBL1728064 0.77 HTR4 (0.59) HTR4HTR3ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899324-B1 Benzimidazole-carboxamide compounds as 5-HT4 receptor agonists THERAVANCE INC (US) 2011-11-30 EP claimed