SCHEMBL1728620

SCHEMBL1728620

CC(C)c1nc2c(OC(=O)NCC3CCNCC3)cccc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 13/20 0.49
HTR3A P46098 10/20 0.49
PARP1 P09874 3/20 0.46
CHRM1 P11229 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL828936 0.82 HTR4 (0.68) HTR4HTR3APARP1CHRM1
SCHEMBL29397140 0.82 HTR4 (0.68) HTR4HTR3APARP1CHRM1
SCHEMBL1726614 0.77 HTR4 (0.59) HTR4HTR3A
SCHEMBL1728218 0.77 HTR4 (0.63) HTR4HTR3APARP1
SCHEMBL1727585 0.77 HTR4 (0.59) HTR4HTR3APARP1
Trifluoroacetic Acid SCHEMBL829123 0.77 HTR4 (0.61) HTR4HTR3APARP1CHRM1
Trifluoroacetic Acid SCHEMBL29399435 0.77 HTR4 (0.61) HTR4HTR3APARP1CHRM1
SCHEMBL1728189 0.76 HTR4 (0.59) HTR4HTR3APARP1
SCHEMBL1728064 0.76 HTR4 (0.59) HTR4HTR3A
SCHEMBL828983 0.76 HTR4 (0.82) HTR4HTR3APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1899324-B1 Benzimidazole-carboxamide compounds as 5-HT4 receptor agonists THERAVANCE INC (US) 2011-11-30 EP claimed