Androstenedone

Androstenedone

SCHEMBL172864

C[C@]12C=CC(=O)C=C1CCC1C2CC[C@]2(C)C(=O)CCC12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 17/20 1.00
CYP3A4 P08684 1/20 1.00
LMNA P02545 2/20 0.66
MAPT P10636 2/20 0.66

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Androstenedone SCHEMBL134061 1.00 CYP19A1 (1.00) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL1144460 1.00 CYP19A1 (1.00) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL12430773 1.00 CYP19A1 (1.00) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL3758714 1.00 CYP19A1 (1.00) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL14450072 1.00 CYP19A1 (1.00) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL10597170 0.99 CYP19A1 (0.97) CYP19A1CYP3A4LMNAMAPT
Androstenedone SCHEMBL4266758 0.92 CYP19A1 (0.84) CYP19A1CYP3A4LMNA
SCHEMBL6897786 0.88 CYP19A1 (0.79) CYP19A1CYP3A4LMNAMAPT
SCHEMBL8491921 0.86 CYP19A1 (0.76) CYP19A1CYP3A4LMNA
SCHEMBL6999301 0.86 CYP19A1 (0.76) CYP19A1CYP3A4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2142561-B9 PROCESS FOR PREPARING AROMATASE INHIBITORS SCINOPHARM TAIWAN LTD (TW) 2014-02-19 EP disclosed
US-8541609-B2 Exemestane and its intermediates and methods of making the same CEDARBURG PHARMACEUTICALS, INC. (US) 2013-09-24 US disclosed
EP-2142561-B1 PROCESS FOR PREPARING AROMATASE INHIBITORS SCINOPHARM TAIWAN LTD (TW) 2013-06-26 EP disclosed
EP-1709062-B9 EXEMESTANE AND ITS INTERMEDIATES AND METHODS OF MAKING THE SAME CEDARBURG PHARMACEUTICALS INC (US) 2013-02-13 EP disclosed
US-8288571-B2 Process for preparing aromatiase inhibitor exemestane CADILA HEALTHCARE LIMITED (IN) 2012-10-16 US disclosed
US-8288571-B2 Process for preparing aromatiase inhibitor exemestane CADILA HEALTHCARE LIMITED (IN) 2012-10-16 US disclosed
US-20120209016-A1 Exemestane and its Intermediates and Methods of Making the Same APOLLO ADMINISTRATIVE AGENCY LLC, AS SUCCESSOR AGENT 2012-08-16 US disclosed
US-8183401-B2 Aromatase inhibitor; deprotonation CEDARBURG PHARMACEUTICALS, INC. (US) 2012-05-22 US disclosed
EP-1709062-B1 EXEMESTANE AND ITS INTERMEDIATES AND METHODS OF MAKING THE SAME CEDARBURG PHARMACEUTICALS INC (US) 2012-03-07 EP disclosed
US-20110028711-A1 Unsaturated Steroid Compounds BIOVIE INC. 2011-02-03 US disclosed
US-20080275259-A1 Process for preparing aromatase inhibitors SCINOPHARM TAIWAN, LTD (TW) 2008-11-06 US disclosed
US-20080275259-A1 Process for preparing aromatase inhibitors SCINOPHARM TAIWAN, LTD (TW) 2008-11-06 US disclosed
US-20080234505-A1 Exemestane and Its Intermediates and Methods of Making the Same CEDARBURG PHARMACEUTICALS, INC (US) 2008-09-25 US disclosed
US-20080070881-A1 Prostate Cancer Treatment HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-03-20 US disclosed
US-20080070881-A1 Prostate Cancer Treatment HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-03-20 US disclosed
US-20080009472-A1 Prostate Cancer Treatment HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-01-10 US disclosed
US-20080009472-A1 Prostate Cancer Treatment HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-01-10 US disclosed
US-20080004250-A1 Compounds and Formulations HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-01-03 US disclosed
US-20080004250-A1 Compounds and Formulations HOLLIS-EDEN PHARMACEUTICALS, INC. (US) 2008-01-03 US disclosed
WO-2007041564-A2 (S)-6-METHYLOXAALKYL EXEMESTANE COMPOUNDS AND RELATED METHODS OF USE ENDECE, LLC (US) 2007-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080070881-A1 Prostate Cancer Treatment AR, KLK3, PTGER1 CYP19A1 49/4885CYP3A4 1241/4885LMNA 3897/4885
US-20080275259-A1 Process for preparing aromatase inhibitors CYP19A1, HSD17B11, CYP17A1 CYP19A1 1/4885CYP3A4 22/4885LMNA 1671/4885
US-20080234505-A1 Exemestane and Its Intermediates and Methods of Making the Same CYP19A1, ESR1, CYP21A2 CYP19A1 1/4885CYP3A4 35/4885LMNA 2022/4885
US-20080009472-A1 Prostate Cancer Treatment AR, KLK3, PTGER1 CYP19A1 49/4885CYP3A4 1241/4885LMNA 3897/4885
US-20110028711-A1 Unsaturated Steroid Compounds PTGER1, AR, PTGES3 CYP19A1 35/4885CYP3A4 1126/4885LMNA 2659/4885
US-20120209016-A1 Exemestane and its Intermediates and Methods of Making the Same CYP19A1, ESR1, CYP21A2 CYP19A1 1/4885CYP3A4 35/4885LMNA 2022/4885
US-20080004250-A1 Compounds and Formulations AR, PTGER1, NR5A1 CYP19A1 18/4885CYP3A4 706/4885LMNA 3184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.