SCHEMBL17295176

SCHEMBL17295176

CCOC(=O)CCc1ccc(Br)c(OC)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.55
CYP4A11 Q02928 1/20 0.55
STING1 Q86WV6 2/20 0.49
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
DRD2 P14416 1/20 0.47
ALOX5 P09917 2/20 0.47
OR51E2 Q9H255 1/20 0.47
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP4Z1 Q86W10 1/20 0.45
TNF P01375 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C8 P10632 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2B6 P20813 1/20 0.44
CYP2C19 P33261 1/20 0.44
ABL1 P00519 1/20 0.44
RIN1 Q13671 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4450867 0.89 CYP4F2 (0.55) CYP4F2CYP4A11STING1KMT2AMEN1
SCHEMBL16294204 0.87 ALOX5 (0.54) KMT2AMEN1ALOX5OR51E2LMNA
SCHEMBL491276 0.87 CYP4F2 (0.59) CYP4F2CYP4A11KMT2AMEN1DRD2
SCHEMBL8984891 0.85 CYP4F2 (0.58) CYP4F2CYP4A11KMT2ADRD2ALOX5
SCHEMBL31053236 0.85 ABL1 (0.56) STING1KMT2AMEN1DRD2ALOX5
SCHEMBL15056738 0.85 ABL1 (0.56) STING1KMT2AMEN1DRD2ALOX5
SCHEMBL8912630 0.85 CYP4F2 (0.58) CYP4F2CYP4A11KMT2ADRD2ALOX5
Dihydroferulic Acid Ethyl Ester SCHEMBL356300 0.84 ALOX5 (0.67) CYP4F2CYP4A11ALOX5OR51E2LMNA
SCHEMBL31236982 0.84 ALDH1A1 (0.42) STING1KMT2AMEN1DRD2LMNA
SCHEMBL4167602 0.83 CYP4F2 (0.55) CYP4F2CYP4A11ALOX5OR51E2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed
WO-2015181272-A1 RAB GERANYLGERANYL TRANSFERASE INHIBITORS LEAD DISCOVERY CENTER GMBH (DE) 2015-12-03 WO disclosed