SCHEMBL1733769

SCHEMBL1733769

C=C(C)C(=O)OCCNC(=O)OCCc1ccc(O)c(-n2nc3ccc(Cl)cc3n2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.35
HTT P42858 3/20 0.35
LMNA P02545 3/20 0.35
TSHR P16473 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
EPHX2 P34913 1/20 0.35
MAPT P10636 4/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
HRH4 Q9H3N8 1/20 0.33
HRH3 Q9Y5N1 1/20 0.33
RXFP1 Q9HBX9 1/20 0.32
TP53 P04637 1/20 0.32
MAPK8 P45983 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL105442 0.92 LMNA (0.35) LMNAMAPTMEN1CYP1A2CYP2C9
SCHEMBL29384829 0.92 LMNA (0.35) LMNAMAPTMEN1CYP1A2CYP2C9
SCHEMBL31132214 0.90 LMNA (0.40) MAPK1HTTLMNATSHRL3MBTL1
SCHEMBL7102773 0.90 LMNA (0.40) MAPK1HTTLMNATSHRL3MBTL1
SCHEMBL2775132 0.86 TLR8 (0.34) HTTLMNATSHRMAPTMEN1
SCHEMBL29512642 0.86 TLR8 (0.34) HTTLMNATSHRMAPTMEN1
SCHEMBL30039355 0.82 LMNA (0.36) MAPK1LMNAMAPTMEN1KMT2A
SCHEMBL7268063 0.81 NPC1 (0.46) LMNAL3MBTL1MAPTSMN1; SMN2MEN1
SCHEMBL93485 0.81 NPC1 (0.47) MAPK1LMNAL3MBTL1MAPTSMN1; SMN2
SCHEMBL29358846 0.81 NPC1 (0.47) MAPK1LMNAL3MBTL1MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 29 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811393-B1 SOFT INTRAOCULAR LENS HOYA CORP (JP) 2002-01-23 EP claimed
US-5814680-A COPOLYMER OF PERFLUOROOCTYLETHYLOXYPROPYLENE (METH) ACRYLATE, PHENYLETHYL (METH)ACRYLATE, ALKYL (METH)ACRYLATE, CROSSLINKING MONOMER HOYA CORPORATION (JP) 1998-09-29 US claimed
EP-0811393-A1 SOFT INTRAOCULAR LENS HOYA CORPORATION (JP) 1997-12-10 EP claimed
US-20210292447-A1 POLYMER MATERIAL AND INTRAOCULAR LENS SHANGHAI FULO MEDICAL INSTRUMENT CO., LTD. (CN) 2021-09-23 US disclosed
EP-3805290-A1 POLYMER MATERIAL AND INTRAOCULAR LENS Shanghai Chartwell Medical Instrument Co., Ltd (CN) 2021-04-14 EP disclosed
US-9529119-B2 Method for fabricating silicone-containing copolymer molded article having hydrophilic surface and silicone-hydrogel contact lens having hydrophilic surface HOYA CORPORATION (JP) 2016-12-27 US disclosed
US-20160282516-A1 METHOD FOR FABRICATING SILICONE-CONTAINING COPOLYMER MOLDED ARTICLE HAVING HYDROPHILIC SURFACE AND SILICONE-HYDROGEL CONTACT LENS HAVING HYDROPHILIC SURFACE HOYA CORPORATION (JP) 2016-09-29 US disclosed
EP-2845708-B1 METHOD FOR PRODUCING SILICONE-CONTAINING COPOLYMER MOLDED ARTICLE HAVING HYDROPHILIC SURFACE, AND SILICONE HYDROGEL CONTACT LENS HAVING HYDROPHILIC SURFACE HOYA CORP (JP) 2016-07-06 EP disclosed
US-20150353667-A1 FLEXIBLE, HIGH REFRACTIVE INDEX HYDROPHOBIC COPOLYMER COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2015-12-10 US disclosed
EP-2926967-A1 Silicone hydrogel contact lens having hydrophilic surface HOYA CORPORATION (JP) 2015-10-07 EP disclosed
EP-2845708-A1 METHOD FOR PRODUCING SILICONE-CONTAINING COPOLYMER MOLDED ARTICLE HAVING HYDROPHILIC SURFACE, AND SILICONE HYDROGEL CONTACT LENS HAVING HYDROPHILIC SURFACE HOYA Corporation (JP) 2015-03-11 EP disclosed
US-20020188352-A1 INTRAOCULAR LENSES AND PROCESS FOR THE PRODUCING MOLDED-IN TYPE INTRAOCULAR LENSES HOYA HEALTHCARE CORPORATION (JP) 2002-12-12 US disclosed
EP-0811393-B1 SOFT INTRAOCULAR LENS HOYA CORP (JP) 2002-01-23 EP disclosed
US-20020005933-A1 Materials for contact lenses comprising a macromer having the polysiloxane structure in the side chain HOYA CORPORATION (JP) 2002-01-17 US disclosed
EP-1128191-A2 Materials for contact lenses comprising a macromer having the polysiloxane structure in the side chain HOYA HEALTHCARE CORPORATION (JP) 2001-08-29 EP disclosed
EP-0968727-A1 INTRAOCULAR LENSES AND PROCESS FOR PRODUCING MOLDED-IN TYPE INTRAOCULAR LENSES Hoya Healthcare Corporation (JP) 2000-01-05 EP disclosed
US-5965630-A POLYMERIZING HYDROPHILIC MONOMERS, HYDROXYETHYL METHACRYLATE, VINYL-2-PYRROLIDONE, DIMETHYLACRYLAMIDE, AN ALKYL METHACRYLATE AND A CROSSLINKER IN A DILUENT OF TRIETHYLENE GLYCOL, DI- OR TRIETHYLENE GLYCOL MONOMETHYL ETHER HOYA CORPORATION (JP) 1999-10-12 US disclosed
US-5814680-A COPOLYMER OF PERFLUOROOCTYLETHYLOXYPROPYLENE (METH) ACRYLATE, PHENYLETHYL (METH)ACRYLATE, ALKYL (METH)ACRYLATE, CROSSLINKING MONOMER HOYA CORPORATION (JP) 1998-09-29 US disclosed
EP-0823643-A1 Soft contact lens with high moisture content and method for producing the same HOYA CORPORATION (JP) 1998-02-11 EP disclosed
EP-0811393-A1 SOFT INTRAOCULAR LENS HOYA CORPORATION (JP) 1997-12-10 EP disclosed