SCHEMBL17339192

SCHEMBL17339192

CCOC(=O)c1cc(Cl)c2ccccn12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.56
ALDH1A1 P00352 8/20 0.56
HPGD P15428 5/20 0.56
GAA P10253 3/20 0.56
GLA P06280 1/20 0.56
MAPT P10636 5/20 0.53
L3MBTL1 Q9Y468 4/20 0.53
NPSR1 Q6W5P4 3/20 0.53
RXFP1 Q9HBX9 1/20 0.52
MAPK1 P28482 4/20 0.50
CYP1A2 P05177 2/20 0.50
CYP3A4 P08684 2/20 0.50
IDO1 P14902 1/20 0.50
HBB P68871 1/20 0.50
HIF1A Q16665 1/20 0.50
TDP1 Q9NUW8 2/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
NOD2 Q9HC29 3/20 0.48
NOD1 Q9Y239 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17339205 0.85 KDM4E (0.58) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL17339148 0.82 ALDH1A1 (0.61) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL17339104 0.80 KDM4E (0.52) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL19961539 0.79 FNTA (0.48) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL19726648 0.77 KDM4E (0.56) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL17339178 0.77 FNTA (0.52) KDM4EALDH1A1MAPTIDO1FNTA
SCHEMBL28532373 0.77 ALDH1A1 (0.55) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL17912564 0.77 ALDH1A1 (0.47) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL17912613 0.76 ALDH1A1 (0.49) KDM4EALDH1A1HPGDGAAGLA
SCHEMBL9535179 0.76 KDM4E (0.69) KDM4EALDH1A1HPGDGAAGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892579-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-07-25 CN disclosed
CN-111875585-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-06-23 CN disclosed
CN-111892579-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-06 CN disclosed
CN-111875585-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-03 CN disclosed
CN-106660993-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-09-11 CN disclosed
CN-106660993-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2017-05-10 CN disclosed
WO-2015188777-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO LTD (CN) 2015-12-17 WO disclosed