SCHEMBL17339205

SCHEMBL17339205

CCOC(=O)c1cc(C)c2ccccn12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.58
ALDH1A1 P00352 5/20 0.58
GAA P10253 3/20 0.58
HPGD P15428 3/20 0.58
GLA P06280 1/20 0.58
NPSR1 Q6W5P4 2/20 0.54
RXFP1 Q9HBX9 1/20 0.54
CYP1A2 P05177 3/20 0.49
MAPK1 P28482 2/20 0.49
CYP3A4 P08684 2/20 0.49
IDO1 P14902 1/20 0.49
HBB P68871 1/20 0.49
HIF1A Q16665 1/20 0.49
FNTA P49354 1/20 0.48
FNTB P49356 1/20 0.48
ATM Q13315 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
HTT P42858 1/20 0.48
MAPT P10636 4/20 0.47
TSHR P16473 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17339192 0.85 KDM4E (0.56) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL17339148 0.84 ALDH1A1 (0.61) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL14963083 0.83 KDM4E (0.49) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL17339104 0.82 KDM4E (0.52) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL10362977 0.81 KDM4E (0.82) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL17339062 0.79 FNTA (0.51) KDM4EALDH1A1GLARXFP1FNTA
SCHEMBL7439300 0.79 BAZ2B (0.64) FNTAFNTBMAPT
SCHEMBL28532373 0.79 ALDH1A1 (0.55) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL9535179 0.78 KDM4E (0.69) KDM4EALDH1A1GAAHPGDGLA
SCHEMBL7449672 0.78 BAZ2B (0.46) KDM4EALDH1A1GAAHPGDGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111892579-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-07-25 CN disclosed
CN-111875585-B Kinase inhibitors 上海艾力斯医药科技股份有限公司 2023-06-23 CN disclosed
CN-111892579-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-06 CN disclosed
CN-111875585-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-11-03 CN disclosed
CN-106660993-B Kinase inhibitor 上海复尚慧创医药研究有限公司 2020-09-11 CN disclosed
CN-106660993-A Kinase inhibitor 上海复尚慧创医药研究有限公司 2017-05-10 CN disclosed
WO-2015188777-A1 CERTAIN PROTEIN KINASE INHIBITORS SHANGHAI FOCHON PHARMACEUTICAL CO LTD (CN) 2015-12-17 WO disclosed