SCHEMBL17355137

SCHEMBL17355137

Bc1ccc2c(c1)C(=O)C1(Cc3ccccc3C1)C2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 3/20 0.36
NPSR1 Q6W5P4 3/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HTR2A P28223 3/20 0.34
HTR2C P28335 3/20 0.34
HTR2B P41595 3/20 0.34
SIGMAR1 Q99720 2/20 0.34
TDP1 Q9NUW8 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
PPIB P23284 1/20 0.33
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CES1 P23141 1/20 0.31
MAOA P21397 1/20 0.31
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29620731 0.79 TDP1 (0.56) L3MBTL1TDP1MAPK1CES1
SCHEMBL6794055 0.79 ESR1 (0.44) LMNAALDH1A1MAOA
SCHEMBL1463836 0.79 TDP1 (0.56) L3MBTL1TDP1MAPK1CES1
SCHEMBL6799540 0.76 PPIB (0.58) L3MBTL1NPSR1LMNAALDH1A1HTR2A
SCHEMBL17355125 0.74 BACE1 (0.39) BACE1
SCHEMBL14026041 0.71 MAOA (0.67) L3MBTL1LMNAALDH1A1TDP1SMN1; SMN2
SCHEMBL6794708 0.70 PBRM1 (0.46) MAOA
SCHEMBL1463869 0.70 TDP1 (0.53) L3MBTL1NPSR1HTR2AHTR2CHTR2B
SCHEMBL31599138 0.70 SIGMAR1 (0.51) L3MBTL1NPSR1HTTLMNAPOLB
SCHEMBL11500029 0.70 SIGMAR1 (0.51) L3MBTL1NPSR1HTTLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2406240-B1 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS INC (US) 2015-12-23 EP disclosed