SCHEMBL1734296

SCHEMBL1734296

CCC(CC1CC1)Nc1nc(C(N)=O)cc(-c2ccccc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.48
ADORA1 P30542 5/20 0.45
VCP P55072 9/20 0.44
HTT P42858 2/20 0.43
GLA P06280 2/20 0.43
FPR2 P25090 1/20 0.43
SCN9A Q15858 1/20 0.43
HSD17B10 Q99714 2/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
ADORA3 P0DMS8 2/20 0.42
ADORA2A P29274 2/20 0.42
ADORA2B P29275 1/20 0.42
LMNA P02545 1/20 0.41
POLB P06746 1/20 0.41
GPR55 Q9Y2T6 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1735520 0.89 KDM4E (0.56) KDM4EADORA1HTTGLAFPR2
SCHEMBL1735526 0.88 SCN9A (0.49) KDM4EVCPGLAFPR2SCN9A
SCHEMBL1735530 0.88 ADORA1 (0.46) ADORA1VCPADORA3ADORA2AADORA2B
SCHEMBL1733485 0.87 VCP (0.49) KDM4EADORA1VCPFPR2SCN9A
SCHEMBL1734498 0.84 VCP (0.47) ADORA1VCPFPR2SCN9AALDH1A1
SCHEMBL1734431 0.84 KDM4E (0.51) KDM4EADORA1HTTGLAFPR2
SCHEMBL1734181 0.83 KDM4E (0.50) KDM4EADORA1HTTGLAFPR2
SCHEMBL1733456 0.78 VCP (0.70) VCP
SCHEMBL1733575 0.78 FPR2 (0.55) KDM4EADORA1HTTGLAFPR2
SCHEMBL1734509 0.77 KDM4E (0.49) KDM4EADORA1HTTGLAFPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed