SCHEMBL1735531

SCHEMBL1735531

NC(=O)c1cc(-c2ccccc2)nc(NCCc2ccco2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.45
ALDH1A1 P00352 6/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
NTRK1 P04629 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
VCP P55072 1/20 0.43
POLB P06746 2/20 0.42
HSD17B10 Q99714 2/20 0.42
HTT P42858 2/20 0.42
LMNA P02545 2/20 0.42
GPR55 Q9Y2T6 1/20 0.42
RAB9A P51151 2/20 0.42
MAPK8 P45983 1/20 0.42
HPGD P15428 4/20 0.41
TSHR P16473 3/20 0.41
GAA P10253 1/20 0.41
CASP1 P29466 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734611 0.90 ALDH1A1 (0.52) KDM4EALDH1A1SMN1; SMN2ADORA2AADORA1
SCHEMBL1734521 0.83 HRH1 (0.52) KDM4EALDH1A1SMN1; SMN2ADORA3ADORA2A
SCHEMBL1734127 0.80 KDM4E (0.57) KDM4EALDH1A1SMN1; SMN2ADORA3ADORA2A
SCHEMBL1735729 0.79 KDM4E (0.48) KDM4EALDH1A1SMN1; SMN2VCPPOLB
SCHEMBL1733447 0.79 VCP (0.48) KDM4EALDH1A1SMN1; SMN2ADORA3ADORA2A
SCHEMBL1734608 0.78 ALDH1A1 (0.55) KDM4EALDH1A1SMN1; SMN2POLBHSD17B10
SCHEMBL1734508 0.77 KDM4E (0.46) KDM4EALDH1A1VCPHSD17B10HTT
SCHEMBL1734267 0.77 PIK3CB (0.57) KDM4EALDH1A1SMN1; SMN2ADORA2AVCP
SCHEMBL1734332 0.77 KDM4E (0.60) KDM4EALDH1A1SMN1; SMN2ADORA3ADORA2A
SCHEMBL1734504 0.77 KDM4E (0.51) KDM4EALDH1A1SMN1; SMN2ADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed