SCHEMBL17364403

SCHEMBL17364403

CCCNc1cccc(NCCC)n1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.51
CHRNB4 P30926 3/20 0.51
CHRNA3 P32297 3/20 0.51
CHRNA4 P43681 3/20 0.51
KCNH2 Q12809 2/20 0.47
SCN5A Q14524 2/20 0.47
CACNA1C Q13936 1/20 0.47
APP P05067 5/20 0.44
TLR8 Q9NR97 1/20 0.43
CNR1 P21554 1/20 0.43
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
HCAR3 P49019 1/20 0.42
ALDH1A1 P00352 1/20 0.41
BLM P54132 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
PIM1 P11309 1/20 0.40
PDE5A O76074 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1742293 0.92 APP (0.54) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL23182746 0.87 NPSR1 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL17364384 0.87 CHRNB2 (0.53) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL14432383 0.86 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL24772646 0.86 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL12893079 0.86 CHRNB2 (0.43) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL12893444 0.86 MEN1 (0.49) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL24329605 0.86 CHRNB2 (0.46) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL516003 0.85 TLR8 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2
SCHEMBL513006 0.82 APP (0.43) CHRNB2CHRNB4CHRNA3CHRNA4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9221821-B2 Methods for the synthesis of 1,3-substituted aminouracils and other xanthine-related compounds Forest Laboratories Holdings, Limited (BM) 2015-12-29 US disclosed