SCHEMBL17364384

SCHEMBL17364384

CCCNc1cccc(NCCOC)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 4/20 0.53
CHRNB4 P30926 4/20 0.53
CHRNA3 P32297 4/20 0.53
CHRNA4 P43681 4/20 0.53
CYP1A2 P05177 6/20 0.48
ALDH1A1 P00352 4/20 0.48
CYP2C19 P33261 3/20 0.48
ALOX15 P16050 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
KCNH3 Q9ULD8 1/20 0.45
BLM P54132 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
CLK4 Q9HAZ1 2/20 0.44
GLA P06280 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2D6 P10635 1/20 0.43
CYP3A4 P08684 2/20 0.42
HCAR3 P49019 1/20 0.42
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17365662 0.93 CYP1A2 (0.53) CHRNB2CHRNB4CHRNA3CHRNA4CYP1A2
SCHEMBL17364403 0.87 CHRNB2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL14621975 0.86 APP (0.50) CHRNB2CHRNB4CHRNA3CHRNA4CYP1A2
SCHEMBL29971364 0.82 CYP1A2 (0.48) CYP1A2ALDH1A1CYP2C19ALOX15HIF1A
SCHEMBL22242112 0.82 CYP1A2 (0.51) CHRNB2CHRNB4CHRNA3CHRNA4CYP1A2
SCHEMBL1099062 0.81 NCF1 (0.49) CYP1A2ALDH1A1CYP2C19ALOX15HIF1A
SCHEMBL29265646 0.81 CYP1A2 (0.47) CHRNB2CHRNA4CYP1A2ALDH1A1CYP2C19
SCHEMBL21894334 0.81 CYP1A2 (0.47) CYP1A2ALDH1A1CYP2C19ALOX15HIF1A
SCHEMBL1742293 0.79 APP (0.54) CHRNB2CHRNB4CHRNA3CHRNA4ALDH1A1
SCHEMBL11001236 0.79 GRM5 (0.48) CHRNB2CHRNB4CHRNA3CHRNA4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9221821-B2 Methods for the synthesis of 1,3-substituted aminouracils and other xanthine-related compounds Forest Laboratories Holdings, Limited (BM) 2015-12-29 US disclosed