Maleic Acid

Maleic Acid

SCHEMBL1737647

O=C(O)/C=C\C(=O)O.O=C1CCCN1

nearest known ligand 0.65

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OR51E2 Q9H255 1/20 0.65
CRBN Q96SW2 3/20 0.56
FKBP5 Q13451 1/20 0.56
KDM4E B2RXH2 3/20 0.40
GAA P10253 1/20 0.40
POLB P06746 1/20 0.40
TSHR P16473 2/20 0.39
TP53 P04637 2/20 0.39
EGLN1 Q9GZT9 1/20 0.39
EGLN3 Q9H6Z9 1/20 0.39
ITGB3 P05106 1/20 0.34
ITGB1 P05556 1/20 0.34
ITGAV P06756 1/20 0.34
ITGA4 P13612 1/20 0.34
INMT O95050 3/20 0.34
KMT2A Q03164 2/20 0.33
MAPT P10636 2/20 0.33
BLM P54132 1/20 0.33
HTT P42858 2/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9716900 1.00 OR51E2 (0.65) OR51E2CRBNFKBP5KDM4EGAA
Fumaric Acid SCHEMBL9716897 1.00 OR51E2 (0.65) OR51E2CRBNFKBP5KDM4EGAA
Maleic Acid SCHEMBL11241940 0.94 OR51E2 (0.58) OR51E2CRBNFKBP5KDM4EGAA
Fumaric Acid SCHEMBL11241948 0.94 OR51E2 (0.58) OR51E2CRBNFKBP5KDM4EGAA
2-Pyrrolidone SCHEMBL27434219 0.88 OR51E2 (0.56) OR51E2CRBNFKBP5KDM4EGAA
Monomethyl Fumarate SCHEMBL11316349 0.86 HCAR2 (0.55) OR51E2CRBNFKBP5KDM4EGAA
Monomethyl Fumarate SCHEMBL11316342 0.86 HCAR2 (0.55) OR51E2CRBNFKBP5KDM4EGAA
2-Pyrrolidone SCHEMBL14977810 0.86 OR51E2 (0.79) OR51E2CRBNFKBP5KDM4EGAA
2-Pyrrolidone SCHEMBL353224 0.86 OR51E2 (0.79) OR51E2CRBNFKBP5KDM4EGAA
2-Pyrrolidone SCHEMBL6929736 0.86 OR51E2 (0.79) OR51E2CRBNFKBP5KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106232059-A Inflatable occluding wire balloon for aortic applications 曲瓦斯库勒股份有限公司 2016-12-14 CN disclosed
EP-3042718-A1 DEVICE FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO- OR NANOEMULSIFICATION Dietz, Ulrich (DE) 2016-07-13 EP disclosed
US-20160122686-A1 DEVICE AND METHOD FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO-OR NANOEMULSIFICATION DIETZ ULRICH (DE) 2016-05-05 US disclosed
EP-2585420-B1 METHOD FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO- OR NANOEMULSIFICATION DIETZ ULRICH (DE) 2016-04-06 EP disclosed
US-9127233-B2 Device and method for solubilizing, separating, removing and reacting carboxylic acids in oils, fats, aqueous or organic solutions by means of micro-or nanoemulsification Dietz, Ulrich (DE) 2015-09-08 US disclosed
EP-2585420-A2 DEVICE AND METHOD FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO- OR NANOEMULSIFICATION Dietz, Ulrich (DE) 2013-05-01 EP disclosed
US-20130090488-A1 DEVICE AND METHOD FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO-OR NANOEMULSIFICATION DIETZ ULRICH (DE) 2013-04-11 US disclosed
CN-101849209-B Composition for forming top anti-reflection film and pattern forming method using the same AZ ELECTRONIC MATERIALS JAPAN 2012-11-28 CN disclosed
CN-101568991-B Top anti-reflective coating composition, method of forming pattern, and top anti-reflective coating AZ ELECTRONIC MATERIALS JAPAN 2012-05-30 CN disclosed
WO-2011160857-A2 DEVICE AND METHOD FOR SOLUBILIZING, SEPARATING, REMOVING AND REACTING CARBOXYLIC ACIDS IN OILS, FATS, AQUEOUS OR ORGANIC SOLUTIONS BY MEANS OF MICRO- OR NANOEMULSIFICATION DIETZ ULRICH (DE) 2011-12-29 WO disclosed
EP-2399885-A1 Device and method for solubilizing, separating, removing and reacting carboxylic acids in aqueous or organic solutions by means of micro- or nanoemulsification Dietz, Ulrich (DE) 2011-12-28 EP disclosed
CN-101849209-A Composition for forming top anti-reflection film and pattern forming method using the same AZ ELECTRONIC MATERIALS JAPAN 2010-09-29 CN disclosed
CN-100587600-C Composition for antireflection coating and pattern formation method using the same DAINIPPON INK & CHEMICALS 2010-02-03 CN disclosed
CN-101568991-A Composition for forming antireflection film and pattern forming method using the same AZ ELECTRONIC MATERIALS JAPAN (JP) 2009-10-28 CN disclosed
CN-101031846-A Composition for antireflection coating and pattern formation method using the same DAINIPPON INK & CHEMICALS (JP) 2007-09-05 CN disclosed