SCHEMBL1739261

SCHEMBL1739261

O=C(O)N1CC(Oc2cnccn2)C1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.47
GRIN1 Q05586 2/20 0.47
GRIN2B Q13224 2/20 0.47
CYP2C9 P11712 1/20 0.47
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
FAAH O00519 4/20 0.42
NAAA Q02083 6/20 0.41
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
KDM4E B2RXH2 1/20 0.37
NAPRT Q6XQN6 1/20 0.37
HCAR2 Q8TDS4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20137677 0.88 EPHX2 (0.55) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL20137678 0.88 EPHX2 (0.55) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL5266581 0.85 EPHX2 (0.60) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL20958357 0.80 NAAA (0.53) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL2997553 0.80 GPR119 (0.52) EPHX2GRIN1GRIN2BCYP2C9NAAA
SCHEMBL1740359 0.78 EPHX2 (0.50) EPHX2FAAH
SCHEMBL14874081 0.77 CHRM2 (0.49) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL20958461 0.77 NAAA (0.51) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL20958463 0.77 NAAA (0.51) EPHX2GRIN1GRIN2BCYP2C9CHRM2
SCHEMBL20958462 0.77 NAAA (0.51) EPHX2GRIN1GRIN2BCYP2C9CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2389382-A1 Amino-heterocyclic compounds used as pde9 inhibitors Pfizer Inc. (US) 2011-11-30 EP disclosed
US-8041687-B2 Dynamic generation of XML Schema for backend driven data validation INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2011-10-18 US disclosed
WO-2010084438-A1 AMINO-HETEROCYCLIC COMPOUNDS USED AS PDE9 INHIBITORS PFIZER INC. (US) 2010-07-29 WO disclosed