SCHEMBL1740468

SCHEMBL1740468

Nc1nc2nc[nH]c2c(=O)n1C(=O)N(c1ccccc1)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 2/20 0.40
ENPP1 P22413 1/20 0.37
BRAF P15056 1/20 0.37
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
TSHR P16473 2/20 0.36
CYP1A2 P05177 2/20 0.36
CDK2 P24941 2/20 0.36
LMNA P02545 1/20 0.36
CDK1 P06493 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CCNB1 P14635 1/20 0.36
MGMT P16455 1/20 0.36
NFKB1 P19838 1/20 0.36
CCNA2 P20248 1/20 0.36
CYP2C19 P33261 1/20 0.36
BLM P54132 1/20 0.36
CCNA1 P78396 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5694191 0.81 NPC1 (0.51) PNPENPP1ALDH1A1TSHRCYP1A2
SCHEMBL1740456 0.81 ALDH1A1 (0.36) PNPALDH1A1MAPK1TSHRCYP1A2
Benzene SCHEMBL8024450 0.79 MGMT (0.43) PNPENPP1ALDH1A1CYP1A2CDK2
SCHEMBL22319176 0.79 PIK3CD (0.36) MAPK1PIK3CD
SCHEMBL28368763 0.78 PNP (0.45) PNPENPP1ALDH1A1TSHRCYP1A2
SCHEMBL6821773 0.77 PNP (0.45) PNPALDH1A1CYP1A2CDK2LMNA
SCHEMBL25398225 0.76 LMNA (0.53) PNPENPP1ALDH1A1MAPK1TSHR
SCHEMBL5694108 0.76 MEN1 (0.41) PNPENPP1TSHRCYP1A2CDK2
SCHEMBL218669 0.76 MGMT (0.45) PNPALDH1A1CYP1A2CDK2CDK1
SCHEMBL29131185 0.76 CDK2 (0.38) PNPENPP1BRAFCDK2CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399588-A1 Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Merck Sharp & Dohme Corp. (US) 2011-12-28 EP disclosed
EP-2360166-A1 Nucleoside derivatives as inhibitors of RNA-dependent RNA viral polymerase Merck Sharp & Dohme Corp. (US) 2011-08-24 EP disclosed
EP-1539188-A2 NUCLEOSIDE DERIVATIVES AS INHIBITORS OF RNA-DEPENDENT RNA VIRAL POLYMERASE Merck & Co., Inc. (US) 2005-06-15 EP disclosed
WO-2002057425-A2 NUCLEOSIDE DERIVATIVES AS INHIBITORS OF RNA-DEPENDENT RNA VIRAL POLYMERASE MERCK & CO., INC. (US) 2002-07-25 WO disclosed
EP-0648220-A1 DEUTERATED NUCLEOSIDES CHATTOPADHYAYA, Jyoti (SE) 1995-04-19 EP disclosed
EP-0421739-A1 3'-azido purine nucleoside THE WELLCOME FOUNDATION LIMITED (GB) 1991-04-10 EP disclosed