SCHEMBL1740550

SCHEMBL1740550

O=C(O)N1CC(c2ncc(Cl)cn2)C1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 6/20 0.48
SCD O00767 1/20 0.37
SCD5 Q86SK9 1/20 0.37
HRH4 Q9H3N8 1/20 0.35
HDAC4 P56524 2/20 0.33
PROKR1 Q8TCW9 3/20 0.33
GRM5 P41594 1/20 0.33
AOC3 Q16853 1/20 0.32
NPC1 O15118 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
SPR P35270 1/20 0.32
PDE9A O76083 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2636853 0.87 HSD11B1 (0.60) HSD11B1AOC3NPC1LMNATP53
SCHEMBL1742207 0.82 HSD11B1 (0.41) HSD11B1HDAC4PROKR1NPC1TP53
SCHEMBL25295913 0.82 HDAC4 (0.36) HSD11B1HDAC4NPC1MAPTRAB9A
SCHEMBL1740546 0.79 PDE10A (0.40) SCDSCD5LMNA
SCHEMBL31622418 0.79 HSD11B1 (0.39) HSD11B1SCD5HRH4HDAC4SPR
SCHEMBL23211853 0.78 SCD5 (0.45) HSD11B1SCDSCD5PROKR1GRM5
SCHEMBL25298297 0.77 FASN (0.42) PROKR1
SCHEMBL25255898 0.76 SCD5 (0.38) HSD11B1SCDSCD5PROKR1NPC1
SCHEMBL162009 0.71 NAPRT (0.43) SMN1; SMN2
SCHEMBL23453444 0.70 SMN1; SMN2 (0.49) HSD11B1PROKR1NPC1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2389382-A1 Amino-heterocyclic compounds used as pde9 inhibitors Pfizer Inc. (US) 2011-11-30 EP disclosed
US-8041687-B2 Dynamic generation of XML Schema for backend driven data validation INTERNATIONAL BUSINESS MACHINES CORPORATION (US) 2011-10-18 US disclosed
WO-2010084438-A1 AMINO-HETEROCYCLIC COMPOUNDS USED AS PDE9 INHIBITORS PFIZER INC. (US) 2010-07-29 WO disclosed