SCHEMBL17409809

SCHEMBL17409809

COCCC1Cc2ccc(C)cc2C1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
CYP19A1 P11511 2/20 0.37
FYN P06241 1/20 0.37
SGPL1 O95470 1/20 0.36
S1PR1 P21453 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
ACHE P22303 1/20 0.34
METAP1 P53582 2/20 0.32
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
MCHR1 Q99705 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
CYP26A1 O43174 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13313179 0.80 IDO1 (0.63) IDO1CYP19A1DRD3
SCHEMBL25080856 0.79 FYN (0.39) IDO1CYP19A1FYNACHEMETAP1
SCHEMBL25818510 0.76 METAP1 (0.41) FYNCHRM2CHRM1CHRM3ACHE
SCHEMBL11532857 0.76 ACHE (0.39) CYP19A1FYNACHEMETAP1MCHR1
SCHEMBL31683941 0.76 ACHE (0.39) CYP19A1FYNACHEMETAP1MCHR1
SCHEMBL30492694 0.74 TRPM5 (0.42) CYP19A1FYNACHEMETAP1
SCHEMBL20584776 0.74 TRPM5 (0.42) CYP19A1FYNACHEMETAP1
SCHEMBL23555197 0.72 ACHE (0.39) IDO1CHRM2CHRM1CHRM3ACHE
SCHEMBL13291785 0.71 MCHR1 (0.39) ACHEMETAP1MCHR1
SCHEMBL10609048 0.70 ACHE (0.39) CYP19A1ACHEMETAP1MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9433622-B2 Pyrimidine compounds useful in the treatment of diseases mediated by IKKE and/or TBK1 mechanisms CASE WESTERN RESERVE UNIVERSITY (US) 2016-09-06 US disclosed
US-20160000784-A1 PYRIMIDINE COMPOUNDS USEFUL IN THE TREATMENT OF DISEASES MEDIATED BY IKKE AND/OR TBK1 MECHANISMS DOMAINEX LIMITED (GB) 2016-01-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160000784-A1 PYRIMIDINE COMPOUNDS USEFUL IN THE TREATMENT OF DISEASES MEDIATED BY IKKE AND/OR TBK1 MECHANISMS TBK1, TBKBP1, TYMS IDO1 1001/4885CYP19A1 4399/4885FYN 1427/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.