SCHEMBL17410230

SCHEMBL17410230

Bc1csc(C(=O)OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTPS1 P17812 1/20 0.42
DAO P14920 1/20 0.39
MAPT P10636 3/20 0.39
NPSR1 Q6W5P4 4/20 0.38
LMNA P02545 2/20 0.38
PPARG P37231 1/20 0.38
NCOA2 Q15596 1/20 0.38
NCOA1 Q15788 1/20 0.38
NCOA3 Q9Y6Q9 1/20 0.38
HPGD P15428 4/20 0.37
ALDH1A1 P00352 4/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPK1 P28482 3/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CA12 O43570 2/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10125215 0.79
SCHEMBL161928 0.78 CTPS1 (0.43) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL294584 0.78 CA12 (0.47) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL70248 0.78 CA1 (0.47) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL1529765 0.78 CES2 (0.59) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL131369 0.78 DAO (0.67) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL14047757 0.77
SCHEMBL25399448 0.76 OPRD1 (0.45) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL19638255 0.76 CTPS1 (0.49) CTPS1DAOMAPTNPSR1LMNA
SCHEMBL21713056 0.76 CES2 (0.57) CTPS1DAOMAPTNPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3517112-B1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME MILLENNIUM PHARM INC (US) 2021-04-07 EP disclosed
WO-2016004136-A1 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME DUFFEY MATTHEW O (US) 2016-01-07 WO disclosed