SCHEMBL25399448

SCHEMBL25399448

COC(=O)c1cc(OC)cs1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CTPS1 P17812 1/20 0.42
MAPT P10636 4/20 0.41
KDM4E B2RXH2 4/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
RAB9A P51151 2/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HPGD P15428 3/20 0.41
CYP3A4 P08684 1/20 0.41
LMNA P02545 3/20 0.40
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HSD17B10 Q99714 1/20 0.40
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4703482 0.86 DAO (0.55) CA1CA2MAPTKDM4EGLA
SCHEMBL28147113 0.83 MEN1 (0.39) CA2MAPTL3MBTL1RAB9AALDH1A1
SCHEMBL7031481 0.83 CTPS1 (0.39) OPRD1CA1CA2CTPS1MAPT
SCHEMBL27953727 0.82 CTPS1 (0.39) OPRD1CA1CA2CTPS1MAPT
SCHEMBL26998951 0.82 CTPS1 (0.39) OPRD1CA1CA2CTPS1MAPT
SCHEMBL8627970 0.82 HPGD (0.47) CA1CA2MAPTKDM4EL3MBTL1
SCHEMBL18302448 0.82 MAPT (0.52) MAPTKDM4EL3MBTL1RAB9AHPGD
SCHEMBL25399545 0.80 KMT2A (0.54) CA1CA2MAPTATMHPGD
SCHEMBL3055932 0.80 MEN1 (0.37) CA2MAPTKDM4EL3MBTL1RAB9A
SCHEMBL6881198 0.79 OPRD1 (0.56) OPRD1CA1CA2MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. 2023-11-16 US disclosed
CN-116490507-A Heterocyclic condensation CDC7 kinase inhibitors for the treatment of cancer 薛定谔公司 2023-07-25 CN disclosed
EP-4211140-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER Schrödinger, Inc. (US) 2023-07-19 EP disclosed
WO-2022055963-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER SCHRÖDINGER, INC. (US) 2022-03-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230365584-A1 HETEROCYCLIC PERICONDENSED CDC7 KINASE INHIBITORS FOR THE TREATMENT OF CANCER CDC7, BUB1B, CDK7 OPRD1 4375/4885CA1 3661/4885CA2 3234/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.