SCHEMBL17416615

SCHEMBL17416615

CCc1c(OC(=O)NN(C(=O)c2cc(C)cc(C)c2)C(CC)C(C)(C)C)ccc2c1OCCO2

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 3/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 3/20 0.34
TP53 P04637 2/20 0.34
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
NPC1 O15118 1/20 0.32
GLA P06280 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GAA P10253 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17416648 0.94 ABCB1 (0.34) ABCB1CYP3A4MAPTTP53HSD17B10
SCHEMBL17416589 0.91 MAPT (0.35) ABCB1CYP3A4MAPTTP53RXFP1
SCHEMBL17416594 0.91 PLK1 (0.36) MAPTTP53MAPK1HSD17B10NPC1
SCHEMBL17416646 0.85 ABCB1 (0.32) ABCB1CYP3A4MAPTTP53HSD17B10
SCHEMBL17416622 0.85 PLK1 (0.35) MAPTTP53MAPK1NPC1RAB9A
SCHEMBL29684694 0.85 ABCB1 (0.39) ABCB1CYP3A4MAPTUSP2ALOX15
SCHEMBL667409 0.85 ABCB1 (0.39) ABCB1CYP3A4MAPTUSP2ALOX15
SCHEMBL12841128 0.83 ABCB1 (0.36) ABCB1CYP3A4MAPTUSP2ALOX15
SCHEMBL29685124 0.79 ABCB1 (0.38) ABCB1CYP3A4MAPTNPC1RAB9A
SCHEMBL668095 0.79 ABCB1 (0.38) ABCB1CYP3A4MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2460786-B1 Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex INTREXON CORP (US) 2016-01-13 EP claimed