SCHEMBL174473

SCHEMBL174473

COc1ccc(F)cc1NC(=O)Nc1cccc2c1CCN2

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 7/20 0.55
KMT2A Q03164 7/20 0.55
MAPT P10636 5/20 0.55
HTT P42858 1/20 0.55
ALDH1A1 P00352 3/20 0.45
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
GAA P10253 1/20 0.43
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
SENP6 Q9GZR1 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
IGF1R P08069 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173758 0.88 SMN1; SMN2 (0.53) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL167730 0.87 MEN1 (0.57) MEN1KMT2AMAPTALDH1A1KDM4E
Trifluoroacetic Acid SCHEMBL167491 0.83 KMT2A (0.50) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL15077842 0.80 IGF1R (0.48) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL175118 0.80 RAB9A (0.58) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL27807412 0.78 MAPT (0.51) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL175262 0.77 SMN1; SMN2 (0.55) MEN1KMT2AMAPTKDM4ESMN1; SMN2
Trifluoroacetic Acid SCHEMBL165260 0.76 IGF1R (0.44) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL174238 0.74 DDX3X (0.52) MEN1KMT2AMAPTHTTALDH1A1
SCHEMBL4569778 0.73 MEN1 (0.53) MEN1KMT2AMAPTHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611806-A1 DEUTERIUM-ENRICHED HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Ascepion Pharmaceuticals, Inc. (CN) 2013-07-10 EP disclosed
WO-2012028106-A1 DEUTERIUM-ENRICHED HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS ASCEPION PHARMACEUTICALS, INC. (CN) 2012-03-08 WO disclosed