SCHEMBL17467968

SCHEMBL17467968

Cc1c(C(N)=O)cnc2cc(C(F)(F)F)cnc12

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.42
SYK P43405 1/20 0.42
PARP1 P09874 3/20 0.41
AGBL2 Q5U5Z8 1/20 0.41
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39
CSF1R P07333 1/20 0.39
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
NNMT P40261 3/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C19 P33261 1/20 0.37
SLC2A1 P11166 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15738937 0.87 AGBL2 (0.46) AGBL2POLBPKMALDH1A1KDM4E
SCHEMBL27855175 0.79 CSF1R (0.51) KMT2ASYKPARP1CSF1R
SCHEMBL17467966 0.71 CSF1R (0.39) SYKCSF1RNNMT
SCHEMBL15922616 0.70 SMN1; SMN2 (0.53) KMT2AAGBL2ALDH1A1KDM4EMAPT
SCHEMBL16666657 0.70 KMT2A (0.50) KMT2ASYKPARP1AGBL2ALDH1A1
SCHEMBL1865699 0.70 SMN1; SMN2 (0.53) KMT2ASYKPARP1AGBL2ALDH1A1
SCHEMBL11159389 0.70 PARP1 (0.54) KMT2ASYKPARP1CSF1RALDH1A1
SCHEMBL15862919 0.69 KMT2A (0.49) KMT2ASYKPARP1AGBL2ALDH1A1
SCHEMBL30056948 0.69 CASP1 (0.52) KMT2AALDH1A1MAPTSMN1; SMN2GAA
SCHEMBL2634210 0.69 CASP1 (0.52) KMT2AALDH1A1MAPTSMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9248122-B2 Heteroquinoline-3-carboxamides as KCNQ2/3 modulators Grünenthal GmbH (DE) 2016-02-02 US disclosed