SCHEMBL17469797

SCHEMBL17469797

Cn1cc(-c2ccc(NNc3c(N)ncc4ccc(Br)cc34)cc2)cn1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CCNC P24863 8/20 0.45
CDK8 P49336 8/20 0.45
AXL P30530 2/20 0.41
LRRK2 Q5S007 2/20 0.41
MET P08581 2/20 0.39
AURKB Q96GD4 1/20 0.39
GSK3B P49841 1/20 0.38
DYRK1A Q13627 1/20 0.38
MAP4K4 O95819 1/20 0.38
IKBKE Q14164 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
ACVR1 Q04771 1/20 0.38
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469719 0.77 KIT (0.59) CCNCCDK8AXLLRRK2MET
SCHEMBL17469641 0.73 KIT (0.47) MAPK1
SCHEMBL17469656 0.72 KIT (0.43)
SCHEMBL25419916 0.71 LRRK2 (0.52) CCNCCDK8LRRK2METAURKB
SCHEMBL20916078 0.69 MET (0.49) CCNCCDK8LRRK2METAURKB
SCHEMBL31165753 0.69 MET (0.49) CCNCCDK8LRRK2METAURKB
SCHEMBL967870 0.69 KCNH2 (0.54) CCNCCDK8AXLLRRK2ACVR1
SCHEMBL19532040 0.66 KIT (0.46)
SCHEMBL30003784 0.66 KIT (0.46)
SCHEMBL25427609 0.65 LRRK2 (0.49) CCNCCDK8LRRK2AURKBGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014674-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2016-01-28 WO disclosed