SCHEMBL17469641

SCHEMBL17469641

N=C(NO)c1ccc(NNc2c(N)ncc3ccc(Br)cc23)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.47
FLT3 P36888 1/20 0.47
NTRK3 Q16288 1/20 0.47
F2 P00734 1/20 0.33
HDAC3 O15379 1/20 0.33
APP P05067 1/20 0.33
ACHE P22303 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
PLG P00747 1/20 0.32
PLAU P00749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469656 0.88 KIT (0.43) KITFLT3NTRK3F2
SCHEMBL17469662 0.85 KIT (0.40) KITFLT3NTRK3F2HDAC3
SCHEMBL21103816 0.77 KIT (0.47) KITFLT3NTRK3HDAC1HDAC6
SCHEMBL17469655 0.76 KIT (0.79) KITFLT3NTRK3F2PLG
SCHEMBL17469797 0.73 CCNC (0.45) MAPK1
SCHEMBL17469875 0.69 FLT3 (0.41) KITFLT3NTRK3F2
SCHEMBL17469644 0.67 FLT3 (0.78) KITFLT3NTRK3F2PLG
SCHEMBL24503717 0.66 KIT (0.48) KITFLT3NTRK3ACHEPLG
SCHEMBL17469637 0.65 KIT (0.72) KITFLT3NTRK3F2PLG
SCHEMBL17469778 0.65 KIT (0.70) KITFLT3NTRK3PLGPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016014674-A1 LINKED DIARYL COMPOUNDS WITH ANTICANCER PROPERTIES AND METHODS OF USING THE SAME UNIVERSITY OF MARYLAND, COLLEGE PARK (US) 2016-01-28 WO disclosed