SCHEMBL1748104

SCHEMBL1748104

CC(C)Oc1cc(CN2CCC(c3ncc(N)c(N)n3)CC2)cc(OC(C)C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 1/20 0.45
ALDH1A1 P00352 2/20 0.39
CCR5 P51681 3/20 0.37
PDE2A O00408 2/20 0.35
FAAH O00519 2/20 0.35
DHFR P00374 1/20 0.35
MAP3K12 Q12852 1/20 0.34
ROCK1 Q13464 1/20 0.33
GMNN O75496 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
DRD2 P14416 1/20 0.33
HPGD P15428 1/20 0.33
DRD4 P21917 1/20 0.33
DRD3 P35462 1/20 0.33
PMP22 Q01453 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1877448 0.82 SSTR5 (0.42) SSTR5ALDH1A1CCR5PDE2AFAAH
SCHEMBL4050604 0.76 SSTR5 (0.47) SSTR5ALDH1A1CCR5PDE2AFAAH
SCHEMBL1748632 0.74 ALDH1A1 (0.50) SSTR5ALDH1A1FAAHGMNNLMNA
SCHEMBL28775007 0.72 FAAH (0.49) SSTR5ALDH1A1CCR5PDE2AFAAH
SCHEMBL27733028 0.71 SSTR5 (0.48) SSTR5ALDH1A1PDE2AFAAHGMNN
SCHEMBL3772265 0.70 SSTR5 (0.50) SSTR5ALDH1A1
SCHEMBL3782674 0.68 SSTR5 (0.60) SSTR5ALDH1A1FAAHGMNNLMNA
SCHEMBL3779040 0.68 SSTR5 (0.55) SSTR5ALDH1A1FAAHROCK2
SCHEMBL1875837 0.68 SSTR5 (0.37) SSTR5ALDH1A1CCR5
SCHEMBL27769482 0.68 ALDH1A1 (0.52) SSTR5ALDH1A1FAAHLMNADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044054-B1 PYRIMIDINE AND QUINAZOLINE DERIVATIVES AS MODULATORS OF SOMATOSTATINE RECEPTOR ACTIVITY HOFFMANN LA ROCHE (CH) 2011-06-08 EP disclosed