SCHEMBL17486014

SCHEMBL17486014

FC(F)(F)c1cc(-c2ccc3c(c2)C2CCC3C2)ncc1Br

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 8/20 0.36
SIGMAR1 Q99720 1/20 0.35
CHRNB2 P17787 2/20 0.35
CHRNA4 P43681 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
KDM1A O60341 3/20 0.33
RPS6KB1 P23443 1/20 0.33
AKT1 P31749 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17486041 0.85 NOTUM (0.41) NOTUMSIGMAR1CHRNB2CHRNA4CHRNB4
SCHEMBL17486126 0.84 KDM1A (0.33) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17485995 0.80 GRM5 (0.34) NOTUMSIGMAR1CHRNB2CHRNA4KDM1A
SCHEMBL15615049 0.77 SIGMAR1 (0.33) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL19295169 0.76 IRAK4 (0.38) NOTUMSIGMAR1KDM1ARPS6KB1IRAK4
SCHEMBL20805808 0.76 NOTUM (0.37) NOTUMSIGMAR1KDM1AIRAK4PDE3B
SCHEMBL19295095 0.76 NOTUM (0.35) NOTUMSIGMAR1IRAK4PDE3BPDE3A
SCHEMBL16905416 0.76 ALOX5AP (0.34) SIGMAR1CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL19295072 0.75 HSD17B1 (0.34) KDM1AMAOB
SCHEMBL19295170 0.75 SIGMAR1 (0.35) NOTUMSIGMAR1CHRNB2CHRNA4CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174890-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-03-13 EP disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-9853228-B2 Metal complexes MERCK PATENT GMBH (DE) 2017-12-26 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
US-20170250353-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2017-08-31 US disclosed
WO-2016015815-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2016-02-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170250353-A1 METAL COMPLEXES SOD1, AP1M1, AP3M1 NOTUM 3335/4885SIGMAR1 4317/4885CHRNB2 2266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.