SCHEMBL175199

SCHEMBL175199

O=C(Nc1ccccc1Br)Nc1cccc2c1CCN2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
LMNA P02545 1/20 0.51
CXCR1 P25024 8/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
CASP3 P42574 1/20 0.46
SENP8 Q96LD8 1/20 0.46
SENP7 Q9BQF6 1/20 0.46
SENP6 Q9GZR1 1/20 0.46
CXCR2 P25025 10/20 0.44
ALDH1A1 P00352 1/20 0.44
ADRB3 P13945 1/20 0.43
TSPO P30536 1/20 0.43
SLC6A3 Q01959 1/20 0.43
GRIK1 P39086 1/20 0.42
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4569778 0.84 MEN1 (0.53) HTTMEN1KMT2ARAB9ANPC1
SCHEMBL174936 0.84 MEN1 (0.51) HTTMEN1KMT2ARAB9ANPC1
SCHEMBL174238 0.83 DDX3X (0.52) HTTMEN1KMT2ARAB9ANPC1
SCHEMBL173846 0.82 STING1 (0.53) HTTMEN1KMT2ARAB9ANPC1
SCHEMBL175017 0.81 GAA (0.56) MEN1KMT2AGAACXCR2ALDH1A1
SCHEMBL257377 0.81 GAA (0.45) RAB9ANPC1GAAMAPTALDH1A1
SCHEMBL173758 0.80 SMN1; SMN2 (0.53) HTTMEN1KMT2ARAB9ANPC1
SCHEMBL173797 0.80 MEN1 (0.54) MEN1KMT2ARAB9ANPC1LMNA
SCHEMBL174930 0.78 RAB9A (0.52) MEN1KMT2ARAB9ANPC1GAA
SCHEMBL174986 0.76 KMT2A (0.52) MEN1KMT2ARAB9ANPC1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611806-A1 DEUTERIUM-ENRICHED HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS Ascepion Pharmaceuticals, Inc. (CN) 2013-07-10 EP claimed
WO-2012028106-A1 DEUTERIUM-ENRICHED HETEROCYCLIC COMPOUNDS AS KINASE INHIBITORS ASCEPION PHARMACEUTICALS, INC. (CN) 2012-03-08 WO claimed