SCHEMBL17524601

SCHEMBL17524601

O[n+]1ccc2cccc(Oc3cccc(C(F)(F)F)c3)c2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43
MAPT P10636 3/20 0.42
ABCG2 Q9UNQ0 1/20 0.42
L3MBTL1 Q9Y468 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ICAM1 P05362 1/20 0.39
SELE P16581 1/20 0.39
EPAS1 Q99814 1/20 0.39
ADORA2A P29274 1/20 0.39
F10 P00742 1/20 0.38
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17508487 0.85 BCHE (0.43) BCHEACHEMAPTABCG2L3MBTL1
SCHEMBL17508472 0.74 HPGD (0.47) MAPTABCG2L3MBTL1NPSR1CYP1A2
SCHEMBL8941708 0.70 AR (0.54) MAPTABCG2L3MBTL1NPSR1CYP1A2
SCHEMBL9798371 0.70 LTA4H (0.54) MAPTABCG2L3MBTL1NPSR1CYP1A2
SCHEMBL11960608 0.70 ACHE (0.62) BCHEACHE
SCHEMBL6791603 0.69 RXFP1 (0.58) CYP2C19THRATHRBKDM4EALDH1A1
SCHEMBL30775042 0.69 RXFP1 (0.58) CYP2C19THRATHRBKDM4EALDH1A1
SCHEMBL9546526 0.69 L3MBTL1 (0.55) ABCG2L3MBTL1NPSR1CYP1A2CYP2C9
SCHEMBL9590802 0.68 AR (0.51) MAPTABCG2L3MBTL1NPSR1CYP1A2
SCHEMBL9589393 0.68 AR (0.51) MAPTABCG2L3MBTL1NPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016021742-A1 HETEROCYCLIC COMPOUNDS AS EP4 RECEPTOR ANTAGONISTS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2016-02-11 WO disclosed