SCHEMBL17524945

SCHEMBL17524945

CC(C)(C)OC(=O)NCc1cnc2c(c1)C1(CCN(c3ccc(N)cn3)CC1)C(=O)N2COCC[Si](C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RET P07949 12/20 0.34
MAPK8 P45983 1/20 0.32
CKS1B P61024 1/20 0.32
SKP1 P63208 1/20 0.32
SKP2 Q13309 1/20 0.32
USP7 Q93009 1/20 0.32
KLKB1 P03952 1/20 0.32
KLK1 P06870 1/20 0.32
DGAT1 O75907 1/20 0.31
DYRK1A Q13627 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CACNA1G O43497 1/20 0.31
CACNA1H O95180 1/20 0.31
CACNA1I Q9P0X4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15699763 0.73 NAMPT (0.37)
SCHEMBL17524871 0.72 OPRM1 (0.33)
SCHEMBL27308006 0.68 AOC3 (0.51) CKS1BSKP1SKP2L3MBTL1CACNA1G
SCHEMBL28367574 0.65 PSMB8 (0.39)
SCHEMBL25315913 0.64 ESR2 (0.39)
SCHEMBL30506821 0.64 ESR2 (0.39)
SCHEMBL27037015 0.64 DRD2 (0.58) RET
SCHEMBL23957794 0.64 KLKB1 (0.45) KLKB1KLK1DYRK1AL3MBTL1
SCHEMBL31436447 0.64 DDR1 (0.41) MAPK8
SCHEMBL25317620 0.64 DDR1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed