SCHEMBL17524871

SCHEMBL17524871

COc1cnc2c(c1)C1(CCN(c3ccc(N)cc3)CC1)C(=O)N2COCC[Si](C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.33
DHFR P00374 1/20 0.33
OPRL1 P41146 2/20 0.33
TGFBR1 P36897 2/20 0.32
OPRK1 P41145 1/20 0.32
FYN P06241 1/20 0.32
CYP19A1 P11511 1/20 0.32
ACVR1 Q04771 3/20 0.31
ALDH1A1 P00352 2/20 0.31
ALOX15 P16050 1/20 0.31
MAPT P10636 4/20 0.31
NR1I2 O75469 1/20 0.31
AHR P35869 1/20 0.31
KDM4E B2RXH2 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
RIPK2 O43353 2/20 0.31
NOD2 Q9HC29 2/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SOAT1 P35610 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524917 0.89 EGLN1 (0.33)
SCHEMBL17506487 0.86 NPC1 (0.34) OPRL1OPRK1ALDH1A1MAPTGAA
SCHEMBL17525045 0.84 EGLN1 (0.41) OPRL1
SCHEMBL21912460 0.74 NPC1 (0.30)
SCHEMBL21912465 0.74 DGAT1 (0.31)
SCHEMBL17525046 0.73 OPRL1 (0.35) OPRL1
SCHEMBL15699637 0.73 CALCRL (0.31) OPRK1
SCHEMBL17524945 0.72 RET (0.34)
SCHEMBL18181139 0.70 EGLN1 (0.39) OPRM1OPRL1OPRK1
SCHEMBL17506429 0.70 GAA (0.37) MAPTSMN1; SMN2GAAHSD17B10KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed