SCHEMBL17525993

SCHEMBL17525993

CCOc1c(F)c(F)cc2[nH]c(-c3cccc(C)n3)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CBFB Q13951 8/20 0.51
BTK Q06187 1/20 0.35
F10 P00742 1/20 0.35
PLG P00747 1/20 0.35
PLAU P00749 1/20 0.35
ALDH1A1 P00352 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HPGD P15428 1/20 0.34
ALOX15 P16050 1/20 0.34
CYP2C19 P33261 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CCR1 P32246 1/20 0.34
CCR8 P51685 1/20 0.34
MGAM O43451 2/20 0.34
GAA P10253 2/20 0.34
SI P14410 2/20 0.34
MGAM2 Q2M2H8 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17525998 0.69 BTK (0.44) CBFBBTKALDH1A1TP53CYP3A4
SCHEMBL19230477 0.69 CBFB (0.47) CBFBCCR1CCR8MGAMGAA
SCHEMBL124333 0.68 CBFB (1.00) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL17525994 0.68 CBFB (0.42) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL124235 0.65 CBFB (0.68) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL179154 0.65 CBFB (0.72) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL17525999 0.63 CBFB (0.40) CBFBALDH1A1TP53CYP3A4CYP2D6
SCHEMBL29484635 0.62 NPC1 (0.60) ALDH1A1TP53CYP3A4CYP2D6HPGD
SCHEMBL11570157 0.62 NPC1 (0.60) ALDH1A1TP53CYP3A4CYP2D6HPGD
SCHEMBL21976942 0.62 METAP2 (0.67) CBFBALDH1A1TP53HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016025744-A1 CANCER THERAPEUTICS UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2016-02-18 WO disclosed