SCHEMBL17530211

SCHEMBL17530211

COc1cccc(C2CCN(C(=O)NC(CC(C)C)C(N)=O)CC2)c1

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.56
PRKG1 Q13976 2/20 0.56
CHRM4 P08173 1/20 0.50
DRD2 P14416 3/20 0.49
POLB P06746 2/20 0.47
CTSK P43235 1/20 0.43
USP5 P45974 1/20 0.43
HCRTR2 O43614 1/20 0.43
PDE4B Q07343 1/20 0.43
CCR1 P32246 1/20 0.43
CCR2 P41597 1/20 0.42
EPHX2 P34913 1/20 0.42
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17530252 0.85 CTSS (0.53) ROCK2PRKG1CHRM4DRD2CTSK
Hydrochloric Acid SCHEMBL30206729 0.77 DRD2 (0.56) ROCK2PRKG1CHRM4DRD2USP5
SCHEMBL17530195 0.77 PLK4 (0.47) PRKG1
SCHEMBL17530199 0.76 CTSS (0.48) DRD2CTSK
SCHEMBL2637036 0.74 DRD2 (0.59) ROCK2PRKG1CHRM4DRD2USP5
SCHEMBL14590572 0.74 QDPR (0.61) ROCK2PRKG1CHRM4DRD2USP5
SCHEMBL7659138 0.73 DRD2 (0.69) CHRM4DRD2USP5CCR2
SCHEMBL17529983 0.73 CTSS (0.57) ROCK2PRKG1CHRM4POLBCTSK
SCHEMBL27382202 0.72 DRD2 (0.57) ROCK2PRKG1CHRM4DRD2USP5
Hydrochloric Acid SCHEMBL11816492 0.72 DRD2 (0.61) ROCK2PRKG1CHRM4DRD2USP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027284-A2 PIPERIDINE UREAS AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed