SCHEMBL17530784

SCHEMBL17530784

Cc1cc2cc(C(C)Nc3ncnc(N)n3)c(N3CCN(C(=O)CO)CC3)nc2cc1F

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.35
KCNH2 Q12809 1/20 0.35
OPRK1 P41145 2/20 0.34
KIT P10721 4/20 0.33
SYK P43405 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
SMO Q99835 1/20 0.33
ALK Q9UM73 2/20 0.32
PIK3CD O00329 2/20 0.32
IDH1 O75874 1/20 0.32
AKT1 P31749 1/20 0.31
AKT1S1 Q96B36 1/20 0.31
CDK4 P11802 1/20 0.31
CDK6 Q00534 1/20 0.31
KRAS P01116 1/20 0.31
P2RY12 Q9H244 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL713286 0.84 CDK2 (0.36) CDK2KCNH2OPRK1KITSYK
SCHEMBL713285 0.84 CDK2 (0.36) CDK2KCNH2OPRK1KITSYK
SCHEMBL17530799 0.84 OPRK1 (0.38) OPRK1AKT1
SCHEMBL17530810 0.80 AKT1 (0.45) OPRK1AKT1KRAS
SCHEMBL17530857 0.79 IDH1 (0.34) OPRK1PIK3CDIDH1
SCHEMBL715221 0.78 KIT (0.39) KCNH2KITTRPV1PIK3CDAKT1
SCHEMBL17530778 0.77 ALDH1A1 (0.37) OPRK1TRPV1IDH1KRAS
SCHEMBL17530766 0.77 MAP4K4 (0.40) OPRK1PIK3CDAKT1
SCHEMBL15899831 0.75 PIK3CD (0.39) TRPV1PIK3CD
SCHEMBL17530794 0.75 KIT (0.35) OPRK1KITPIK3CDIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2403847-B1 TRIAZINE DERIVATIVES AS KINASE INHIBITORS UCB BIOPHARMA SPRL (BE) 2016-03-02 EP claimed