SCHEMBL17533593

SCHEMBL17533593

CC(C)(F)CC(NC(=O)c1ccc2c(ccn2S(C)(=O)=O)c1)C(=O)NC1(C#N)CC1

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.48
CTSB P07858 10/20 0.48
CTSL P07711 9/20 0.48
CTSS P25774 8/20 0.48
CTSV O60911 1/20 0.48
CTSF Q9UBX1 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17533671 0.87 CTSL (0.60) CTSKCTSBCTSLCTSS
SCHEMBL17533591 0.85 CTSL (0.60) CTSKCTSBCTSLCTSSCTSF
SCHEMBL17533612 0.72 CTSL (0.61) CTSKCTSBCTSLCTSSCTSV
SCHEMBL17514231 0.72 CTSL (0.57) CTSKCTSBCTSLCTSS
SCHEMBL17533710 0.71 CTSL (0.59) CTSKCTSBCTSLCTSS
SCHEMBL17533636 0.71 CTSL (0.58) CTSKCTSBCTSLCTSS
SCHEMBL17533699 0.71 CTSL (0.58) CTSKCTSBCTSLCTSS
SCHEMBL17533640 0.69 CTSL (0.50) CTSKCTSBCTSLCTSS
SCHEMBL17533579 0.69 PPARG (0.44) CTSKCTSBCTSLCTSS
SCHEMBL17514263 0.69 GRN (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027285-A2 BICYCLIC HETEROARYL AMIDES AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed