SCHEMBL17533591

SCHEMBL17533591

CC(C)(F)CC(NC(=O)c1ccc2c(ccn2S(C)(=O)=O)c1)C(=O)NCC#N

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSL P07711 14/20 0.60
CTSB P07858 8/20 0.44
CTSF Q9UBX1 1/20 0.44
PPARG P37231 3/20 0.43
CTSS P25774 7/20 0.43
CTSK P43235 5/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17533612 0.86 CTSL (0.61) CTSLCTSBCTSSCTSK
SCHEMBL17514231 0.86 CTSL (0.57) CTSLCTSBCTSSCTSK
SCHEMBL17533593 0.85 CTSK (0.48) CTSLCTSBCTSFCTSSCTSK
SCHEMBL17533710 0.84 CTSL (0.59) CTSLCTSBPPARGCTSSCTSK
SCHEMBL17533579 0.82 PPARG (0.44) CTSLCTSBPPARGCTSSCTSK
SCHEMBL17533638 0.78 CTSL (0.56) CTSLCTSBPPARGCTSSCTSK
SCHEMBL17533642 0.76 CTSL (0.53) CTSLCTSBCTSSCTSK
SCHEMBL17514263 0.74 GRN (0.54) PPARG
SCHEMBL17533634 0.74 PPARG (0.38) PPARG
SCHEMBL17533607 0.73 RORC (0.47) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027285-A2 BICYCLIC HETEROARYL AMIDES AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed