SCHEMBL17533671

SCHEMBL17533671

CC(C)CC(NC(=O)c1ccc2c(ccn2S(C)(=O)=O)c1)C(=O)NC1(C#N)CC1

nearest known ligand 0.60

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CTSL P07711 19/20 0.60
CTSS P25774 11/20 0.59
CTSK P43235 11/20 0.59
CTSB P07858 4/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17533593 0.87 CTSK (0.48) CTSLCTSSCTSKCTSB
SCHEMBL17514231 0.84 CTSL (0.57) CTSLCTSSCTSKCTSB
SCHEMBL17533636 0.83 CTSL (0.58) CTSLCTSSCTSKCTSB
SCHEMBL17533699 0.83 CTSL (0.58) CTSLCTSSCTSKCTSB
SCHEMBL17514263 0.81 GRN (0.54)
SCHEMBL17514265 0.78 TAS1R3 (0.47)
SCHEMBL17533641 0.77 CTSL (0.66) CTSLCTSSCTSKCTSB
SCHEMBL17533638 0.76 CTSL (0.56) CTSLCTSSCTSKCTSB
SCHEMBL17533642 0.76 CTSL (0.53) CTSLCTSSCTSKCTSB
SCHEMBL17533710 0.73 CTSL (0.59) CTSLCTSSCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027285-A2 BICYCLIC HETEROARYL AMIDES AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed