SCHEMBL1753613

SCHEMBL1753613

CNS(=O)(=O)c1ccc(-c2cc(Cl)ccc2O[C@@H](C)C(=O)O)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.52
HTR2A P28223 1/20 0.52
HTR2C P28335 1/20 0.52
HTR2B P41595 1/20 0.52
PTGDR2 Q9Y5Y4 6/20 0.48
NLRP3 Q96P20 1/20 0.46
GAA P10253 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA3 P07451 1/20 0.46
CA4 P22748 1/20 0.46
CA6 P23280 1/20 0.46
CA5A P35218 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA13 Q8N1Q1 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CA5B Q9Y2D0 1/20 0.46
MMP2 P08253 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1753455 0.86 PTGDR2 (0.57) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1753537 0.85 PTGDR2 (0.67) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1690331 0.84 TSHR (0.55) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1991361 0.83 TSHR (0.51) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1753812 0.80 ALDH1A1 (0.53) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1753809 0.78 MEN1 (0.56) TSHRPTGDR2GAA
SCHEMBL2100973 0.77 ABCB11 (0.58) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL5186851 0.77 ABCB11 (0.58) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL2111712 0.76 TSHR (0.54) TSHRHTR2AHTR2CHTR2BPTGDR2
SCHEMBL1753451 0.75 PTGDR2 (0.66) TSHRHTR2AHTR2CHTR2BPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8158820-B2 Compounds ASTRAZENECA AB (SE) 2012-04-17 US disclosed