SCHEMBL17537657

SCHEMBL17537657

O=C(c1nc(-c2c[nH]c3ccccc23)cs1)c1c[nH]c2ccccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 8/20 0.63
MEN1 O00255 7/20 0.63
MAPT P10636 6/20 0.63
NR1I2 O75469 1/20 0.62
AHR P35869 1/20 0.62
RAB9A P51151 3/20 0.59
SMN1; SMN2 Q16637 3/20 0.59
ALDH1A1 P00352 3/20 0.59
KDM4E B2RXH2 2/20 0.59
THRB P10828 2/20 0.59
ALOX15 P16050 1/20 0.59
PPARG P37231 1/20 0.59
NCOA2 Q15596 1/20 0.59
HSD17B10 Q99714 1/20 0.59
GPR84 Q9NQS5 1/20 0.55
CGAS Q8N884 1/20 0.55
TDP1 Q9NUW8 2/20 0.54
ATP4A P20648 2/20 0.54
ATP4B P51164 2/20 0.54
AR P10275 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21366458 0.86 MEN1 (0.62) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL21366050 0.84 MAPT (0.60) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL21366246 0.83 MAPT (0.58) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL21366326 0.83 MAPT (0.58) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL21366075 0.83 MAPT (0.58) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL17537647 0.83 ADRA1A (0.50) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL17537643 0.83 NR4A2 (0.47) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL17537646 0.83 ATP4A (0.46) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL21366112 0.82 MAPT (0.57) KMT2AMEN1MAPTNR1I2AHR
SCHEMBL22462583 0.82 MAPT (0.66) KMT2AMEN1MAPTNR1I2AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016023106-A1 BIS-INDOLE ALKALOIDS FOR USE IN THE TREATMENT OF INFECTIONS THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2016-02-18 WO disclosed