SCHEMBL1754933

SCHEMBL1754933

c1ccc(CCC2CCC(Oc3ccc4cnccc4c3)CC2)cc1

nearest known ligand 0.57

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK1 Q13464 8/20 0.57
ROCK2 O75116 3/20 0.57
IKBKB O14920 4/20 0.52
PRKCZ Q05513 1/20 0.51
CCR2 P41597 1/20 0.42
CHUK O15111 3/20 0.41
PRMT3 O60678 1/20 0.41
LCK P06239 1/20 0.41
MRGPRX4 Q96LA9 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
DRD3 P35462 1/20 0.38
KCNH2 Q12809 1/20 0.37
IMPDH2 P12268 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1754919 0.96 ROCK1 (0.53) ROCK1ROCK2IKBKBPRKCZCCR2
SCHEMBL1754935 0.84 IKBKB (0.46) ROCK1ROCK2IKBKBPRKCZCHUK
SCHEMBL1705194 0.83 ROCK1 (0.54) ROCK1ROCK2IKBKBPRKCZCCR2
SCHEMBL1705741 0.83 ROCK1 (0.54) ROCK1ROCK2IKBKBPRKCZCCR2
SCHEMBL1705000 0.83 ROCK1 (0.54) ROCK1ROCK2IKBKBPRKCZCCR2
SCHEMBL1705714 0.81 IKBKB (0.54) ROCK1ROCK2IKBKBPRKCZCHUK
SCHEMBL1705260 0.81 IKBKB (0.54) ROCK1ROCK2IKBKBPRKCZCHUK
SCHEMBL12192827 0.79 ROCK1 (0.76) ROCK1ROCK2IKBKBPRKCZCCR2
SCHEMBL1754929 0.78 LMNA (0.43) ROCK1ROCK2IKBKBPRKCZPRMT3
SCHEMBL1705239 0.78 ROCK1 (0.57) ROCK1ROCK2IKBKBPRKCZCCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125746-B1 CYCLOALKYLAMINE SUBSTITUTED ISOQUINOLINE DERIVATIVES SANOFI SA (FR) 2012-04-18 EP disclosed