SCHEMBL1754929

SCHEMBL1754929

CC1(c2ccc(CCC3CCC(Oc4ccc5cnccc5c4)CC3)cc2)NC(=O)NC1=O

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
IKBKB O14920 1/20 0.43
PRKCZ Q05513 1/20 0.42
ROCK1 Q13464 3/20 0.41
MMP13 P45452 6/20 0.40
ADAM17 P78536 2/20 0.39
ROCK2 O75116 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
MMP14 P50281 3/20 0.37
PRMT3 O60678 2/20 0.34
MMP12 P39900 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704777 0.85 LMNA (0.43) LMNAIKBKBPRKCZROCK1MMP13
SCHEMBL1754933 0.78 ROCK1 (0.57) IKBKBPRKCZROCK1ROCK2PRMT3
SCHEMBL1754935 0.78 IKBKB (0.46) IKBKBPRKCZROCK1ROCK2PRMT3
SCHEMBL1754919 0.77 ROCK1 (0.53) IKBKBPRKCZROCK1ROCK2PRMT3
SCHEMBL1092530 0.74 LMNA (0.54) LMNAMMP13ADAM17MEN1KMT2A
SCHEMBL1705714 0.70 IKBKB (0.54) IKBKBPRKCZROCK1ROCK2PRMT3
SCHEMBL1705260 0.70 IKBKB (0.54) IKBKBPRKCZROCK1ROCK2PRMT3
SCHEMBL1704728 0.67 IKBKB (0.62) IKBKBPRKCZROCK1ROCK2
SCHEMBL102335 0.66 MMP13 (0.44) LMNAMMP13MEN1KMT2AMMP14
SCHEMBL30824363 0.66 ROCK1 (0.72) IKBKBPRKCZROCK1ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2125746-B1 CYCLOALKYLAMINE SUBSTITUTED ISOQUINOLINE DERIVATIVES SANOFI SA (FR) 2012-04-18 EP disclosed